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| Title | Structural snapshots capture nucleotide release at the mu-opioid receptor |
|---|---|
| Journal, issue, pages | Nature, Year 2025 |
| Publish date | Aug 6, 2025 (structure data deposition date) |
Authors | Khan S / Tyson AS / Ranjbar M / Zhang Z / Singh J / Han GW / Gati C |
External links | Nature / Search PubMed |
| Methods | EM (single particle) |
| Resolution | 2.73 - 8.78 Å |
| Structure data | ![]() EMDB-71976: Inactive-state naloxone-mu opioid receptor nanobody6 complex - Consensus map ![]() EMDB-71977: Inactive-state naloxone-mu opioid receptor nanobody6 complex - Locally refined receptor map ![]() EMDB-71978: Inactive-state naloxone-mu opioid receptor nanobody6 complex - Locally refined fiducal map ![]() EMDB-71979: Nucleotide-free naloxone-mu opioid receptor Gi1 complex - Consensus map ![]() EMDB-71980: Nucleotide-free naloxone-mu opioid receptor Gi1 complex - Locally refined receptor map ![]() EMDB-71981: Nucleotide-free naloxone-mu opioid receptor Gi1 complex - Locally refined Gi map ![]() EMDB-71982: Latent-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Consensus map ![]() EMDB-71983: Latent-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined receptor map ![]() EMDB-71984: Latent-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined Gi map ![]() EMDB-71985: Unlatched-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Consensus map ![]() EMDB-71986: Unlatched-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined receptor map ![]() EMDB-71987: Unlatched-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined Gi map ![]() EMDB-71988: Primed-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Consensus map ![]() EMDB-71989: Primed-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined receptor map ![]() EMDB-71990: Primed-state naloxone-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined Gi map ![]() EMDB-71991: Engaged-state loperamide-mu opioid receptor-Gi GDPbS complex (rebound) - Consensus map ![]() EMDB-71992: Engaged-state loperamide-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined receptor map ![]() EMDB-71993: Engaged-state loperamide-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined Gi map ![]() EMDB-71998: Primed-state loperamide-mu opioid receptor-Gi GDPbS complex (rebound) - Consensus map ![]() EMDB-71999: Primed-state loperamide-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined receptor map ![]() EMDB-72000: Primed-state loperamide-mu opioid receptor-Gi GDPbS complex (rebound) - Locally refined Gi GDP map EMDB-72001, PDB-9pxu: EMDB-72002, PDB-9pxv: EMDB-72003, PDB-9pxw: EMDB-72004, PDB-9pxx: EMDB-72005, PDB-9pxy: EMDB-72006, PDB-9py2: EMDB-72008, PDB-9py4: ![]() EMDB-72022: Latent-state loperamide-mu opioid receptor-Gi GDP complex (constant GDP) - Consensus map ![]() EMDB-72023: Latent-state loperamide-mu opioid receptor-Gi GDP complex (constant GDP) - Locally refined map ![]() EMDB-72024: Engaged-state loperamide-mu opioid receptor-Gi GDP complex (constant GDP) - Consensus map ![]() EMDB-72025: Engaged-state loperamide-mu opioid receptor-Gi GDP complex (constant GDP) - Locally refined map ![]() EMDB-72026: Open-AHD loperamide-mu opioid receptor-Gi GDP complex (constant GDP) - Consensus map ![]() EMDB-72027: Open-AHD loperamide-mu opioid receptor-Gi GDP complex (constant GDP) - Locally refined receptor map |
| Chemicals | ![]() PDB-1apv: ![]() ChemComp-NA: ![]() ChemComp-CLR: ![]() ChemComp-VSN: ![]() PDB-1cmv: |
| Source |
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Keywords | MEMBRANE PROTEIN / G protein coupled receptor / Mu Opioid receptor / Naloxone / GDP / Loperamide |
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