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-Structure paper
Title | Discovery of a selective c-MET inhibitor with a novel binding mode. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 75, Page 128948-128948, Year 2022 |
Publish date | Aug 4, 2022 (structure data deposition date) |
Authors | Collie, G.W. / Barlind, L. / Bazzaz, S. / Borjesson, U. / Dale, I.L. / Disch, J.S. / Habeshian, S. / Jetson, R. / Khurana, P. / Madin, A. ...Collie, G.W. / Barlind, L. / Bazzaz, S. / Borjesson, U. / Dale, I.L. / Disch, J.S. / Habeshian, S. / Jetson, R. / Khurana, P. / Madin, A. / Michaelides, I.N. / Peng, L. / Snijder, A. / Stubbs, C.J. |
External links | Bioorg. Med. Chem. Lett. / PubMed:35987508 |
Methods | X-ray diffraction |
Resolution | 2.01 - 2.394 Å |
Structure data | PDB-8an8: PDB-8ans: |
Chemicals | ChemComp-SO4: ChemComp-MDI: ChemComp-HOH: ChemComp-GOL: |
Source |
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Keywords | TRANSFERASE / kinase / inhibitor / aC-helix / cancer |