|
eF-site ID
|
6qfl-A |
PDB Code
|
6qfl |
Chain
|
A |
|
click to enlarge
|
|
Title
|
Structure of the mitogen activated kinase kinase 7 active conformation |
Classification
|
TRANSFERASE |
Compound
|
Dual specificity mitogen-activated protein kinase kinase 7 |
Source
|
(MP2K7_HUMAN) |
|
Sequence
|
A: |
QTGYLTIGGQRYQAEINDLENLGEMGSGTCGQVWKMRFRK
TGHVIAVKQMRRSGNKEENKRILMDLDVVLKSHDCPYIVQ
CFGTFITNTDVFIAMELMGTCAEKLKKRMQGPIPERILGK
MTVAIVKALYYLKEKHGVIHRDVKPSNILLDERGQIKLCD
FGISGRLAGCAAYMAPERIDPPDYDIRADVWSLGISLVEL
ATGQFPYKNCKTDFEVLTKVLQEEPPLLPGHMGFSGDFQS
FVKDCLTKDHRKRPKYNKLLEHSFIKRYETLEVDVASWFK
DVMAKTE
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
A |
residue |
142 |
type |
BINDING |
sequence |
M
|
description |
BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
2)
|
chain |
A |
residue |
165 |
type |
BINDING |
sequence |
K
|
description |
BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
3)
|
chain |
A |
residue |
259 |
type |
ACT_SITE |
sequence |
D
|
description |
Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00159, ECO:0000255|PROSITE-ProRule:PRU10027
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
4)
|
chain |
A |
residue |
255-267 |
type |
prosite |
sequence |
VIHRDVKPSNILL
|
description |
PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. ViHrDVKpsNILL
|
source |
prosite : PS00108
|
|
|
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