eF-site ID 6oqn-B
PDB Code 6oqn
Chain B

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Title Crystal structure of Mcl1 with inhibitor 7
Classification APOPTOSIS
Compound Induced myeloid leukemia cell differentiation protein Mcl-1
Source (MCL1_HUMAN)
Sequence B:  EDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKAL
ETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVM
IHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPL
AESITDVLVRTKRDWLVKQRGWDGFVEFFHV
Description


Functional site

1) chain B
residue 227
type
sequence A
description binding site for residue N0P B 401
source : AC2

2) chain B
residue 249
type
sequence V
description binding site for residue N0P B 401
source : AC2

3) chain B
residue 250
type
sequence M
description binding site for residue N0P B 401
source : AC2

4) chain B
residue 263
type
sequence R
description binding site for residue N0P B 401
source : AC2

5) chain B
residue 266
type
sequence T
description binding site for residue N0P B 401
source : AC2

6) chain B
residue 267
type
sequence L
description binding site for residue N0P B 401
source : AC2

7) chain B
residue 270
type
sequence F
description binding site for residue N0P B 401
source : AC2

8) chain B
residue 290
type
sequence L
description binding site for residue N0P B 401
source : AC2

9) chain B
residue 194
type CROSSLNK
sequence K
description Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
source Swiss-Prot : SWS_FT_FI1

10) chain B
residue 197
type CROSSLNK
sequence K
description Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
source Swiss-Prot : SWS_FT_FI1


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