eF-site ID 6ohu-A
PDB Code 6ohu
Chain A

click to enlarge
Title Structure of EBP and tamoxifen
Classification membrane protein, isomerase/inhibitor
Compound 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase
Source (EBP_HUMAN)
Sequence A:  PLHPYWPQHLRLDNFVPNDRPTWHILAGLFSVTGVLVVTT
WLLSGRTWRRLSLCWFAVCGFIHLVIEGWFVLYYEDLLGD
QAFLSQLWKEYAKGDSRYILGDNFTVCMETITACLWGPLS
LWVVIAFLRQHPLRFILQLVVSVGQIYGDVLYFLTEHRDG
FQHGELGHPLYFWFYFVFMNALWLVLPGVLVLDAVKHLTH
AQSTLD
Description


Functional site

1) chain A
residue 35
type
sequence L
description binding site for residue CTX A 301
source : AC1

2) chain A
residue 36
type
sequence F
description binding site for residue CTX A 301
source : AC1

3) chain A
residue 39
type
sequence T
description binding site for residue CTX A 301
source : AC1

4) chain A
residue 75
type
sequence I
description binding site for residue CTX A 301
source : AC1

5) chain A
residue 79
type
sequence I
description binding site for residue CTX A 301
source : AC1

6) chain A
residue 80
type
sequence E
description binding site for residue CTX A 301
source : AC1

7) chain A
residue 100
type
sequence L
description binding site for residue CTX A 301
source : AC1

8) chain A
residue 101
type
sequence W
description binding site for residue CTX A 301
source : AC1

9) chain A
residue 188
type
sequence Y
description binding site for residue CTX A 301
source : AC1

10) chain A
residue 192
type
sequence M
description binding site for residue CTX A 301
source : AC1

11) chain A
residue 193
type
sequence N
description binding site for residue CTX A 301
source : AC1

12) chain A
residue 196
type
sequence W
description binding site for residue CTX A 301
source : AC1

13) chain A
residue 29-49
type TRANSMEM
sequence WHILAGLFSVTGVLVVTTWLL
description Helical => ECO:0000255
source Swiss-Prot : SWS_FT_FI1

14) chain A
residue 66-86
type TRANSMEM
sequence LCWFAVCGFIHLVIEGWFVLY
description Helical => ECO:0000255
source Swiss-Prot : SWS_FT_FI1

15) chain A
residue 121-141
type TRANSMEM
sequence METITACLWGPLSLWVVIAFL
description Helical => ECO:0000255
source Swiss-Prot : SWS_FT_FI1

16) chain A
residue 185-205
type TRANSMEM
sequence FWFYFVFMNALWLVLPGVLVL
description Helical => ECO:0000255
source Swiss-Prot : SWS_FT_FI1


Display surface

Download
Links