eF-site ID 6nco-A
PDB Code 6nco
Chain A

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Title Fragment-based Discovery of an apoE4 Stabilizer
Classification LIPID TRANSPORT
Compound Apolipoprotein E
Source (APOE_HUMAN)
Sequence A:  QRWELALGRFWDYLRWVQTLSEQVQEELLSSQVTQELRAL
MDETMKELKAYKSELEEQLTPVAEETRARLSKELQAAQAR
LGADMEDVRGRLVQYRGEVQAMLGQSTEELRVRLASHLRK
LRKRLLRDADDLQKRLAVYQA
Description


Functional site

1) chain A
residue 27
type
sequence E
description binding site for residue KQP A 201
source : AC1

2) chain A
residue 30
type
sequence L
description binding site for residue KQP A 201
source : AC1

3) chain A
residue 31
type
sequence G
description binding site for residue KQP A 201
source : AC1

4) chain A
residue 34
type
sequence W
description binding site for residue KQP A 201
source : AC1

5) chain A
residue 35
type
sequence D
description binding site for residue KQP A 201
source : AC1

6) chain A
residue 131
type
sequence E
description binding site for residue KQP A 201
source : AC1

7) chain A
residue 134
type
sequence R
description binding site for residue KQP A 201
source : AC1

8) chain A
residue 149
type
sequence L
description binding site for residue KQP A 201
source : AC1

9) chain A
residue 153
type
sequence D
description binding site for residue KQP A 201
source : AC1

10) chain A
residue 156
type
sequence Q
description binding site for residue KQP A 201
source : AC1

11) chain A
residue 143
type BINDING
sequence K
description BINDING => ECO:0000269|PubMed:3947350
source Swiss-Prot : SWS_FT_FI1

12) chain A
residue 124
type MOD_RES
sequence A
description Methionine sulfoxide => ECO:0000250|UniProtKB:P08226
source Swiss-Prot : SWS_FT_FI2

13) chain A
residue 128
type MOD_RES
sequence Q
description Phosphoserine; by FAM20C => ECO:0000269|PubMed:26091039, ECO:0007744|PubMed:24275569
source Swiss-Prot : SWS_FT_FI3

14) chain A
residue 74
type CARBOHYD
sequence Y
description N-linked (Glc) (glycation) lysine => ECO:0000269|PubMed:10452964
source Swiss-Prot : SWS_FT_FI5


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