eF-site ID 6g9p-A
PDB Code 6g9p
Chain A

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Title Structural basis for the inhibition of E. coli PBP2
Classification HYDROLASE/ANTIBIOTIC
Compound Peptidoglycan D,D-transpeptidase MrdA
Source (MRDA_ECOLI)
Sequence A:  NRIKLVPIAPSRGIIYDRNGIPLALNRTIYQIEMMPEKVD
NVQQTLDALRSVVDLTDDDIAAFRKERARSHRFTSIPVKT
NLTEVQVARFAVNQYRFPGVEVKGYKRRYYPYGSALTHVI
GYVSKINDKDVERLNNDGKLANYAATHDIGKLGIERYYED
VLHGQTGYEEVEVNNRGRVIRQLKEVPPQAGHDIYLTLDL
KLQQYIETLLAGSRAAVVVTDPRTGGVLALVSTPSYDPNL
FVDGISSKDYSALLNDPNTPLVNRATQGVYPPASTVKPYV
AVSALSAGVITRNTTLFDPGWWQLPGSEKRYRDWKKWGHG
RLNVTRSLEESADTFFYQVAYDMGIDRLSEWMGKFGYGHY
TGIDLAEERSGNMPTREWKQKRFKKPWYQGDTIPVGIGQG
YWTATPIQMSKALMILINDGIVKVPHLLMSTAEDGKQVPW
VQPHEPPVGDIHSGYWELAKDGMYGVANRPNGTAHKYFAS
APYKIAAKSGTAQRDHKLMTAFAPYNNPQVAVAMILENGG
AGPAVGTLMRQILDHIML
Description


Functional site

1) chain A
residue 330
type ACT_SITE
sequence S
description Acyl-ester intermediate => ECO:0000255|HAMAP-Rule:MF_02081, ECO:0000269|PubMed:3148617
source Swiss-Prot : SWS_FT_FI1


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