eF-site ID 6frf-ABCD
PDB Code 6frf
Chain A, B, C, D

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Title Crystal structure of CREBBP bromodomain complexd with PA10
Classification TRANSFERASE
Compound CREB-binding protein
Source (CBP_HUMAN)
Sequence A:  MRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQL
LGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWL
MFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG
B:  IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIP
DYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNN
AWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG
C:  IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIP
DYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNN
AWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL
D:  IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIP
DYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNN
AWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG
Description


Functional site

1) chain A
residue 1109
type
sequence L
description binding site for residue E3T A 1201
source : AC1

2) chain A
residue 1110
type
sequence P
description binding site for residue E3T A 1201
source : AC1

3) chain A
residue 1113
type
sequence Q
description binding site for residue E3T A 1201
source : AC1

4) chain A
residue 1115
type
sequence V
description binding site for residue E3T A 1201
source : AC1

5) chain A
residue 1120
type
sequence L
description binding site for residue E3T A 1201
source : AC1

6) chain A
residue 1168
type
sequence N
description binding site for residue E3T A 1201
source : AC1

7) chain A
residue 1173
type
sequence R
description binding site for residue E3T A 1201
source : AC1

8) chain A
residue 1174
type
sequence V
description binding site for residue E3T A 1201
source : AC1

9) chain B
residue 1109
type
sequence L
description binding site for residue E3T B 1201
source : AC2

10) chain B
residue 1110
type
sequence P
description binding site for residue E3T B 1201
source : AC2

11) chain B
residue 1113
type
sequence Q
description binding site for residue E3T B 1201
source : AC2

12) chain B
residue 1115
type
sequence V
description binding site for residue E3T B 1201
source : AC2

13) chain B
residue 1120
type
sequence L
description binding site for residue E3T B 1201
source : AC2

14) chain B
residue 1168
type
sequence N
description binding site for residue E3T B 1201
source : AC2

15) chain B
residue 1173
type
sequence R
description binding site for residue E3T B 1201
source : AC2

16) chain B
residue 1174
type
sequence V
description binding site for residue E3T B 1201
source : AC2

17) chain B
residue 1177
type
sequence F
description binding site for residue E3T B 1201
source : AC2

18) chain C
residue 1116
type
sequence D
description binding site for residue E3T B 1201
source : AC2

19) chain C
residue 1119
type
sequence L
description binding site for residue E3T B 1201
source : AC2

20) chain D
residue 1175
type
sequence Y
description binding site for residue E3T B 1201
source : AC2

21) chain A
residue 1175
type
sequence Y
description binding site for residue E3T C 1201
source : AC3

22) chain B
residue 1119
type
sequence L
description binding site for residue E3T C 1201
source : AC3

23) chain C
residue 1109
type
sequence L
description binding site for residue E3T C 1201
source : AC3

24) chain C
residue 1110
type
sequence P
description binding site for residue E3T C 1201
source : AC3

25) chain C
residue 1113
type
sequence Q
description binding site for residue E3T C 1201
source : AC3

26) chain C
residue 1115
type
sequence V
description binding site for residue E3T C 1201
source : AC3

27) chain C
residue 1120
type
sequence L
description binding site for residue E3T C 1201
source : AC3

28) chain C
residue 1168
type
sequence N
description binding site for residue E3T C 1201
source : AC3

29) chain C
residue 1173
type
sequence R
description binding site for residue E3T C 1201
source : AC3

30) chain C
residue 1177
type
sequence F
description binding site for residue E3T C 1201
source : AC3

31) chain A
residue 1120
type
sequence L
description binding site for residue E3T D 1201
source : AC4

32) chain D
residue 1110
type
sequence P
description binding site for residue E3T D 1201
source : AC4

33) chain D
residue 1113
type
sequence Q
description binding site for residue E3T D 1201
source : AC4

34) chain D
residue 1115
type
sequence V
description binding site for residue E3T D 1201
source : AC4

35) chain D
residue 1120
type
sequence L
description binding site for residue E3T D 1201
source : AC4

36) chain D
residue 1168
type
sequence N
description binding site for residue E3T D 1201
source : AC4

37) chain D
residue 1173
type
sequence R
description binding site for residue E3T D 1201
source : AC4

38) chain D
residue 1174
type
sequence V
description binding site for residue E3T D 1201
source : AC4

39) chain A
residue 1108-1167
type prosite
sequence SLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQY
QEPWQYVDDVWLMFNNAWLY
description BROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
source prosite : PS00633


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