eF-site ID 6fqo-B
PDB Code 6fqo
Chain B

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Title Crystal structure of CREBBP bromodomain complexd with DT29
Classification TRANSFERASE
Compound CREB-binding protein
Source (CBP_HUMAN)
Sequence B:  SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQ
LLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVW
LMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG
Description


Functional site

1) chain B
residue 1165
type
sequence W
description binding site for residue E2T A 1201
source : AC1

2) chain B
residue 1162
type
sequence N
description binding site for residue EDO A 1202
source : AC2

3) chain B
residue 1165
type
sequence W
description binding site for residue EDO A 1202
source : AC2

4) chain B
residue 1109
type
sequence L
description binding site for residue E2T B 1201
source : AC3

5) chain B
residue 1110
type
sequence P
description binding site for residue E2T B 1201
source : AC3

6) chain B
residue 1113
type
sequence Q
description binding site for residue E2T B 1201
source : AC3

7) chain B
residue 1115
type
sequence V
description binding site for residue E2T B 1201
source : AC3

8) chain B
residue 1120
type
sequence L
description binding site for residue E2T B 1201
source : AC3

9) chain B
residue 1168
type
sequence N
description binding site for residue E2T B 1201
source : AC3

10) chain B
residue 1173
type
sequence R
description binding site for residue E2T B 1201
source : AC3

11) chain B
residue 1159
type
sequence L
description binding site for residue EDO B 1202
source : AC4

12) chain B
residue 1162
type
sequence N
description binding site for residue EDO B 1202
source : AC4

13) chain B
residue 1163
type
sequence N
description binding site for residue EDO B 1202
source : AC4


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