eF-site ID 6fgd-A
PDB Code 6fgd
Chain A

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Title Crystal structure of Gephyrin E domain in complex with Artemether
Classification STRUCTURAL PROTEIN
Compound Gephyrin
Source (GEPH_RAT)
Sequence A:  SPFPLTSMDKAFITVLEMTPVLGTEIINYRDGMGRVLAQD
VYAKDNLPPFPASVKDGYAVRAADGPGDRFIIGESQAGEQ
PTQTVMPGQVMRVTTGAPIPCGADAVVQVEDTELIRESDD
GTEELEVRILVQARPGQDIRPIGHDIKRGECVLAKGTHMG
PSEIGLLATVGVTEVEVNKFPVVAVMSTGNELLNPEDDLL
PGKIRDSNRSTLLATIQEHGYPTINLGIVGDNPDDLLNAL
NEGISRADVIITSGGVSMGEKDYLKQVLDIDLHAQIHFGR
VFMKPGLPTTFATLDIDGVRKIIFALPGNPVSAVVTCNLF
VVPALRKMQGILDPRPTIIKARLSCDVKLDPRPEYHRCIL
TWHHQEPLPWAQSTSRLMSMRSANGLLMLPPKTEQYVELH
KGEVVDVMVIGRL
Description


Functional site

1) chain A
residue 580
type
sequence D
description binding site for residue CA A 802
source : AC2

2) chain A
residue 500
type
sequence V
description binding site for residue PO4 A 803
source : AC3

3) chain A
residue 564
type
sequence R
description binding site for residue PO4 A 803
source : AC3

4) chain A
residue 565
type
sequence A
description binding site for residue PO4 A 803
source : AC3

5) chain A
residue 566
type
sequence D
description binding site for residue PO4 A 803
source : AC3

6) chain A
residue 619
type
sequence K
description binding site for residue PO4 A 803
source : AC3

7) chain A
residue 469
type
sequence C
description binding site for residue ACT A 804
source : AC4

8) chain A
residue 470
type
sequence V
description binding site for residue ACT A 804
source : AC4

9) chain A
residue 651
type
sequence D
description binding site for residue ACT A 805
source : AC5

10) chain A
residue 653
type
sequence R
description binding site for residue ACT A 805
source : AC5

11) chain A
residue 476
type
sequence H
description binding site for residue ACT A 806
source : AC6

12) chain A
residue 477
type
sequence M
description binding site for residue ACT A 806
source : AC6

13) chain A
residue 705
type
sequence S
description binding site for residue ACT A 806
source : AC6

14) chain A
residue 339
type
sequence V
description binding site for residue ACT A 807
source : AC7

15) chain A
residue 618
type
sequence R
description binding site for residue ACT A 807
source : AC7

16) chain A
residue 323
type
sequence L
description binding site for residue ACT A 809
source : AC9

17) chain A
residue 325
type
sequence S
description binding site for residue ACT A 809
source : AC9

18) chain A
residue 600
type
sequence F
description binding site for residue ACT A 809
source : AC9

19) chain A
residue 348
type
sequence R
description binding site for residue ACT A 811
source : AD1

20) chain A
residue 535
type
sequence Q
description binding site for residue ACT A 811
source : AD1

21) chain A
residue 343
type
sequence E
description binding site for residue ACT A 812
source : AD2

22) chain A
residue 353
type
sequence R
description binding site for residue ACT A 812
source : AD2

23) chain A
residue 497
type
sequence K
description binding site for residue ACT A 812
source : AD2

24) chain A
residue 498
type
sequence F
description binding site for residue ACT A 812
source : AD2

25) chain A
residue 342
type
sequence T
description binding site for residue ACT A 813
source : AD3

26) chain A
residue 563
type
sequence S
description binding site for residue ACT A 813
source : AD3

27) chain A
residue 335
type
sequence E
description binding site for residue ACT A 814
source : AD4

28) chain A
residue 336
type
sequence M
description binding site for residue ACT A 814
source : AD4

29) chain A
residue 337
type
sequence T
description binding site for residue ACT A 814
source : AD4

30) chain A
residue 338
type
sequence P
description binding site for residue ACT A 814
source : AD4

31) chain A
residue 618
type
sequence R
description binding site for residue ACT A 814
source : AD4

32) chain A
residue 514
type
sequence E
description binding site for residue ACT A 815
source : AD5

33) chain A
residue 514
type
sequence E
description binding site for residue ACT A 815
source : AD5

34) chain A
residue 613
type
sequence D
description binding site for residue ACT A 816
source : AD6

35) chain A
residue 614
type
sequence I
description binding site for residue ACT A 816
source : AD6

36) chain A
residue 615
type
sequence D
description binding site for residue ACT A 816
source : AD6

37) chain A
residue 616
type
sequence G
description binding site for residue ACT A 816
source : AD6

38) chain A
residue 356
type
sequence A
description binding site for residue ACT A 817
source : AD7

39) chain A
residue 613
type
sequence D
description binding site for residue ACT A 818
source : AD8

40) chain A
residue 616
type
sequence G
description binding site for residue ACT A 818
source : AD8

41) chain A
residue 660
type
sequence R
description binding site for residue ACT A 819
source : AD9

42) chain A
residue 724
type
sequence K
description binding site for residue ACT A 819
source : AD9

43) chain A
residue 725
type
sequence G
description binding site for residue ACT A 819
source : AD9

44) chain A
residue 392
type
sequence E
description binding site for residue ACT A 820
source : AE1

45) chain A
residue 397
type
sequence E
description binding site for residue ACT A 820
source : AE1

46) chain A
residue 399
type
sequence P
description binding site for residue ACT A 820
source : AE1

47) chain A
residue 400
type
sequence T
description binding site for residue ACT A 820
source : AE1

48) chain A
residue 401
type
sequence Q
description binding site for residue ACT A 820
source : AE1

49) chain A
residue 335
type
sequence E
description binding site for residue ACT A 821
source : AE2

50) chain A
residue 386
type
sequence D
description binding site for residue ACT A 821
source : AE2

51) chain A
residue 388
type
sequence F
description binding site for residue ACT A 821
source : AE2

52) chain A
residue 406
type
sequence G
description binding site for residue ACT A 821
source : AE2

53) chain A
residue 418
type
sequence P
description binding site for residue ACT A 822
source : AE3

54) chain A
residue 421
type
sequence A
description binding site for residue ACT A 822
source : AE3

55) chain A
residue 544
type
sequence L
description binding site for residue ACT A 823
source : AE4

56) chain A
residue 560
type
sequence E
description binding site for residue ACT A 823
source : AE4

57) chain A
residue 434
type
sequence R
description binding site for residue ACT A 824
source : AE5

58) chain A
residue 444
type
sequence E
description binding site for residue ACT A 824
source : AE5

59) chain A
residue 651
type
sequence D
description binding site for residue ACT A 824
source : AE5

60) chain A
residue 652
type
sequence P
description binding site for residue ACT A 824
source : AE5

61) chain A
residue 653
type
sequence R
description binding site for residue ACT A 824
source : AE5

62) chain A
residue 658
type
sequence K
description binding site for residue ACT A 825
source : AE6

63) chain A
residue 727
type
sequence V
description binding site for residue ACT A 825
source : AE6

64) chain A
residue 728
type
sequence V
description binding site for residue ACT A 825
source : AE6

65) chain A
residue 729
type
sequence D
description binding site for residue ACT A 825
source : AE6

66) chain A
residue 476
type
sequence H
description binding site for residue ACT A 826
source : AE7

67) chain A
residue 644
type
sequence R
description binding site for residue ACT A 826
source : AE7

68) chain A
residue 373
type
sequence K
description binding site for residue ACT A 827
source : AE8

69) chain A
residue 426
type
sequence Q
description binding site for residue ACT A 827
source : AE8

70) chain A
residue 456
type
sequence D
description binding site for residue ACT A 827
source : AE8

71) chain A
residue 625
type
sequence P
description binding site for residue NA A 828
source : AE9

72) chain A
residue 630
type
sequence S
description binding site for residue NA A 828
source : AE9

73) chain A
residue 414
type
sequence G
description binding site for residue ADP A 829
source : AF1

74) chain A
residue 505
type
sequence S
description binding site for residue ADP A 829
source : AF1

75) chain A
residue 509
type
sequence E
description binding site for residue ADP A 829
source : AF1

76) chain A
residue 510
type
sequence L
description binding site for residue ADP A 829
source : AF1

77) chain A
residue 522
type
sequence I
description binding site for residue ADP A 829
source : AF1

78) chain A
residue 524
type
sequence D
description binding site for residue ADP A 829
source : AF1

79) chain A
residue 525
type
sequence S
description binding site for residue ADP A 829
source : AF1

80) chain A
residue 526
type
sequence N
description binding site for residue ADP A 829
source : AF1

81) chain A
residue 572
type
sequence G
description binding site for residue ADP A 829
source : AF1

82) chain A
residue 573
type
sequence G
description binding site for residue ADP A 829
source : AF1

83) chain A
residue 574
type
sequence V
description binding site for residue ADP A 829
source : AF1

84) chain A
residue 575
type
sequence S
description binding site for residue ADP A 829
source : AF1

85) chain A
residue 580
type
sequence D
description binding site for residue ADP A 829
source : AF1

86) chain A
residue 625
type
sequence P
description binding site for residue ADP A 829
source : AF1

87) chain A
residue 626
type
sequence G
description binding site for residue ADP A 829
source : AF1

88) chain A
residue 627
type
sequence N
description binding site for residue ADP A 829
source : AF1

89) chain A
residue 628
type
sequence P
description binding site for residue ADP A 829
source : AF1

90) chain A
residue 480
type
sequence S
description binding site for residue MPD A 830
source : AF2

91) chain A
residue 484
type
sequence L
description binding site for residue MPD A 830
source : AF2

92) chain A
residue 628
type
sequence P
description binding site for residue MPD A 830
source : AF2

93) chain A
residue 675
type
sequence R
description binding site for residue MPD A 830
source : AF2

94) chain A
residue 326
type
sequence M
description binding site for residue D8Z A 831
source : AF3

95) chain A
residue 327
type
sequence D
description binding site for residue D8Z A 831
source : AF3

96) chain A
residue 330
type
sequence F
description binding site for residue D8Z A 831
source : AF3

97) chain A
residue 637
type
sequence L
description binding site for residue D8Z A 831
source : AF3

98) chain A
residue 653
type
sequence R
description binding site for residue D8Z A 831
source : AF3

99) chain A
residue 656
type
sequence I
description binding site for residue D8Z A 831
source : AF3

100) chain A
residue 711
type
sequence M
description binding site for residue D8Z A 831
source : AF3

101) chain A
residue 731
type
sequence M
description binding site for residue D8Z A 831
source : AF3

102) chain A
residue 575-610
type prosite
sequence SMGEKDYLKQVLDIDLHAQIHFGRVFMKPGLPTTFA
description MOCF_BIOSYNTHESIS_2 Molybdenum cofactor biosynthesis proteins signature 2. SmGekDylkqvLdidlhaqihfgrVfmKPGLPttFA
source prosite : PS01079


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