eF-site ID 6el6-AB
PDB Code 6el6
Chain A, B

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Title Glucocorticoid Receptor in complex with compound 4
Classification SIGNALING PROTEIN
Compound Glucocorticoid receptor
Source Homo sapiens (Human) (NCOA2_HUMAN)
Sequence A:  PTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGR
QMIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMSLMAFALG
WRSYRQSSANLLCFAPDLIINEQRMTLPDMYDQCKHMLYV
SSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEI
RMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVV
ENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNI
KKLLFHQ
B:  ENALLRYLLDKDD
Description


Functional site

1) chain A
residue 541
type
sequence P
description binding site for residue EDO A 801
source : AC1

2) chain A
residue 574
type
sequence A
description binding site for residue EDO A 801
source : AC1

3) chain A
residue 577
type
sequence W
description binding site for residue EDO A 801
source : AC1

4) chain A
residue 603
type
sequence L
description binding site for residue EDO A 801
source : AC1

5) chain A
residue 667
type
sequence K
description binding site for residue EDO A 801
source : AC1

6) chain A
residue 563
type
sequence L
description binding site for residue B9Q A 802
source : AC2

7) chain A
residue 564
type
sequence N
description binding site for residue B9Q A 802
source : AC2

8) chain A
residue 566
type
sequence L
description binding site for residue B9Q A 802
source : AC2

9) chain A
residue 567
type
sequence G
description binding site for residue B9Q A 802
source : AC2

10) chain A
residue 570
type
sequence Q
description binding site for residue B9Q A 802
source : AC2

11) chain A
residue 601
type
sequence M
description binding site for residue B9Q A 802
source : AC2

12) chain A
residue 604
type
sequence M
description binding site for residue B9Q A 802
source : AC2

13) chain A
residue 607
type
sequence A
description binding site for residue B9Q A 802
source : AC2

14) chain A
residue 608
type
sequence L
description binding site for residue B9Q A 802
source : AC2

15) chain A
residue 611
type
sequence R
description binding site for residue B9Q A 802
source : AC2

16) chain A
residue 623
type
sequence F
description binding site for residue B9Q A 802
source : AC2

17) chain A
residue 642
type
sequence Q
description binding site for residue B9Q A 802
source : AC2

18) chain A
residue 646
type
sequence M
description binding site for residue B9Q A 802
source : AC2

19) chain A
residue 735
type
sequence Y
description binding site for residue B9Q A 802
source : AC2

20) chain A
residue 736
type
sequence C
description binding site for residue B9Q A 802
source : AC2

21) chain A
residue 739
type
sequence T
description binding site for residue B9Q A 802
source : AC2

22) chain A
residue 703
type CROSSLNK
sequence K
description Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
source Swiss-Prot : SWS_FT_FI1


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