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eF-site ID
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6e3s-A |
PDB Code
|
6e3s |
Chain
|
A |
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click to enlarge
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Title
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Crystal Structure of the Heterodimeric HIF-2 Complex with Antagonist PT2385 |
Classification
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transcription/transcription inhibitor |
Compound
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Aryl hydrocarbon receptor nuclear translocator |
Source
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(EPAS1_MOUSE) |
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Sequence
|
A: |
ERRRRNKMTAYITELSDMVPTCPDKLTILRMAVSHMKSLL
TDQELKHLILEAADGFLFIVSCETGRVVYVSDSVTPVLNQ
PQSEWFGSTLYDQVHPDDVDKLREQLSTSRRSFICRMRCG
TPHFVVVHCTGYIKAWFCLVAIGRLQTEFISRHNIEGIFT
FVDHRCVATVGYQPQELLGKNIVEFCHPEDQQLLRDSFQQ
VVKLKGQVLSVMFRFRSKTREWLWMRTSSFTFQNPYSDEI
EYIICTNTNV
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Description
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