eF-site ID 6dxk-AB
PDB Code 6dxk
Chain A, B

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Title Glucocorticoid Receptor in complex with Compound 11
Classification TRANSCRIPTION
Compound Glucocorticoid receptor
Source (GCR_HUMAN)
Sequence A:  PTLVSALETIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGR
QVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALG
WRSYRQSSANLLCFAPDLIINEQRMTLPDMYDQCKHMLYV
SSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQALFDAI
RMTYIKELGKAIVKREGNSSQNSQRFYQLTKLLDSMHEVV
ENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNI
KKLLFHQ
B:  PTLVSALETIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGR
QVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALG
WRSYRQSSANLLCFAPDLIINEQRMTLPDMYDQCKHMLYV
SSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQALFDAI
RMTYIKELGKAIVKREGNSSQNSQRFYQLTKLLDSMHEVV
ENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNI
KKLLFHQK
Description


Functional site

1) chain A
residue 560
type
sequence M
description binding site for residue HJ4 A 801
source : AC1

2) chain A
residue 568
type
sequence G
description binding site for residue HJ4 A 801
source : AC1

3) chain A
residue 570
type
sequence Q
description binding site for residue HJ4 A 801
source : AC1

4) chain A
residue 604
type
sequence M
description binding site for residue HJ4 A 801
source : AC1

5) chain A
residue 611
type
sequence R
description binding site for residue HJ4 A 801
source : AC1

6) chain A
residue 623
type
sequence F
description binding site for residue HJ4 A 801
source : AC1

7) chain A
residue 735
type
sequence Y
description binding site for residue HJ4 A 801
source : AC1

8) chain A
residue 736
type
sequence C
description binding site for residue HJ4 A 801
source : AC1

9) chain B
residue 557
type
sequence W
description binding site for residue HJ4 A 801
source : AC1

10) chain A
residue 557
type
sequence W
description binding site for residue HJ4 B 801
source : AC2

11) chain B
residue 563
type
sequence L
description binding site for residue HJ4 B 801
source : AC2

12) chain B
residue 564
type
sequence N
description binding site for residue HJ4 B 801
source : AC2

13) chain B
residue 567
type
sequence G
description binding site for residue HJ4 B 801
source : AC2

14) chain B
residue 570
type
sequence Q
description binding site for residue HJ4 B 801
source : AC2

15) chain B
residue 604
type
sequence M
description binding site for residue HJ4 B 801
source : AC2

16) chain B
residue 611
type
sequence R
description binding site for residue HJ4 B 801
source : AC2

17) chain B
residue 623
type
sequence F
description binding site for residue HJ4 B 801
source : AC2

18) chain B
residue 735
type
sequence Y
description binding site for residue HJ4 B 801
source : AC2

19) chain B
residue 758
type
sequence T
description binding site for residue HJ4 B 801
source : AC2

20) chain A
residue 702
type CROSSLNK
sequence V
description Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
source Swiss-Prot : SWS_FT_FI1

21) chain B
residue 702
type CROSSLNK
sequence V
description Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
source Swiss-Prot : SWS_FT_FI1


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