|
eF-site ID
|
6dgq-B |
PDB Code
|
6dgq |
Chain
|
B |
|
click to enlarge
|
|
Title
|
Crystal Structure of Human PPARgamma Ligand Binding Domain in Complex with CAY10506 |
Classification
|
TRANSCRIPTION/TRANSCRIPTION INHIBITOR |
Compound
|
Peroxisome proliferator-activated receptor gamma |
Source
|
(PPARG_HUMAN) |
|
Sequence
|
B: |
ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSP
FVIYDMNSLMMGEDKIKEVAIRIFQGCQFRSVEAVQEITE
YAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDG
VLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALE
LDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALE
LQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKK
TEHPLLQEIYKDL
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
286 |
type |
BINDING |
sequence |
Q
|
description |
BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
2)
|
chain |
B |
residue |
323 |
type |
BINDING |
sequence |
H
|
description |
BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
3)
|
chain |
B |
residue |
449 |
type |
BINDING |
sequence |
H
|
description |
BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
4)
|
chain |
B |
residue |
473 |
type |
BINDING |
sequence |
Y
|
description |
BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
5)
|
chain |
B |
residue |
224 |
type |
CROSSLNK |
sequence |
K
|
description |
Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
|
|