eF-site ID 6db0-C
PDB Code 6db0
Chain C

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Title N-Terminal bromodomain of Human BRD2 with a Tetrahydroquinoline analogue
Classification Transcription/Inhibitor
Compound Bromodomain-containing protein 2
Source (BRD2_HUMAN)
Sequence C:  TNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLPDYHK
IIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIY
NKPTDDIVLMAQTLEKIFLQKVASMPQ
Description


Functional site

1) chain C
residue 128
type
sequence R
description binding site for residue EPE B 302
source : AC4

2) chain C
residue 129
type
sequence R
description binding site for residue EPE B 302
source : AC4

3) chain C
residue 132
type
sequence N
description binding site for residue EPE B 302
source : AC4

4) chain C
residue 134
type
sequence Y
description binding site for residue EPE B 302
source : AC4

5) chain C
residue 113
type
sequence Y
description binding site for residue EDO C 301
source : AC5

6) chain C
residue 156
type
sequence N
description binding site for residue EDO C 301
source : AC5

7) chain C
residue 84
type MOD_RES
sequence K
description Phosphoserine => ECO:0007744|PubMed:19690332
source Swiss-Prot : SWS_FT_FI2

8) chain C
residue 159
type BINDING
sequence T
description BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
source Swiss-Prot : SWS_FT_FI1


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