eF-site ID 6db0-B
PDB Code 6db0
Chain B

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Title N-Terminal bromodomain of Human BRD2 with a Tetrahydroquinoline analogue
Classification Transcription/Inhibitor
Compound Bromodomain-containing protein 2
Source (BRD2_HUMAN)
Sequence B:  PGRVTNQLQYLHKVVMKALWKHQFAWPFRQPVDAVKLGLP
DYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTN
CYIYNKPTDDIVLMAQTLEKIFLQKVASMPQEEQE
Description


Functional site

1) chain B
residue 94
type
sequence Q
description binding site for residue G3J A 302
source : AC2

2) chain B
residue 97
type
sequence W
description binding site for residue G3J B 301
source : AC3

3) chain B
residue 98
type
sequence P
description binding site for residue G3J B 301
source : AC3

4) chain B
residue 99
type
sequence F
description binding site for residue G3J B 301
source : AC3

5) chain B
residue 108
type
sequence L
description binding site for residue G3J B 301
source : AC3

6) chain B
residue 110
type
sequence L
description binding site for residue G3J B 301
source : AC3

7) chain B
residue 156
type
sequence N
description binding site for residue G3J B 301
source : AC3

8) chain B
residue 162
type
sequence I
description binding site for residue G3J B 301
source : AC3

9) chain B
residue 97
type
sequence W
description binding site for residue EPE B 302
source : AC4

10) chain B
residue 100
type
sequence R
description binding site for residue EPE B 302
source : AC4

11) chain B
residue 84
type MOD_RES
sequence K
description Phosphoserine => ECO:0007744|PubMed:19690332
source Swiss-Prot : SWS_FT_FI2

12) chain B
residue 159
type BINDING
sequence T
description BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
source Swiss-Prot : SWS_FT_FI1


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