eF-site ID 6czw-A
PDB Code 6czw
Chain A

click to enlarge
Title Crystal structure of PT1940 bound to HIF2a-B*:ARNT-B* complex
Classification TRANSCRIPTION
Compound Endothelial PAS domain-containing protein 1
Source (ARNT_HUMAN)
Sequence A:  FKGLDSKTFLSEHSMDMKFTYCDDRITELIGYHPEELLGR
SAYEFYHALDSENMTKSHQNLCTKGQVVSGQYRMLAKHGG
YVWLETQGTVIYNPPQCIMCVNYVLSEIE
Description


Functional site

1) chain A
residue 244
type
sequence F
description binding site for residue FO7 A 401
source : AC1

2) chain A
residue 246
type
sequence S
description binding site for residue FO7 A 401
source : AC1

3) chain A
residue 248
type
sequence H
description binding site for residue FO7 A 401
source : AC1

4) chain A
residue 252
type
sequence M
description binding site for residue FO7 A 401
source : AC1

5) chain A
residue 277
type
sequence A
description binding site for residue FO7 A 401
source : AC1

6) chain A
residue 281
type
sequence Y
description binding site for residue FO7 A 401
source : AC1

7) chain A
residue 289
type
sequence M
description binding site for residue FO7 A 401
source : AC1

8) chain A
residue 292
type
sequence S
description binding site for residue FO7 A 401
source : AC1

9) chain A
residue 293
type
sequence H
description binding site for residue FO7 A 401
source : AC1

10) chain A
residue 296
type
sequence L
description binding site for residue FO7 A 401
source : AC1

11) chain A
residue 302
type
sequence V
description binding site for residue FO7 A 401
source : AC1

12) chain A
residue 304
type
sequence S
description binding site for residue FO7 A 401
source : AC1

13) chain A
residue 307
type
sequence Y
description binding site for residue FO7 A 401
source : AC1

14) chain A
residue 309
type
sequence M
description binding site for residue FO7 A 401
source : AC1

15) chain A
residue 321
type
sequence T
description binding site for residue FO7 A 401
source : AC1

16) chain A
residue 323
type
sequence G
description binding site for residue FO7 A 401
source : AC1

17) chain A
residue 339
type
sequence C
description binding site for residue FO7 A 401
source : AC1

18) chain A
residue 341
type
sequence N
description binding site for residue FO7 A 401
source : AC1


Display surface

Download
Links