eF-site ID 6cxs-C
PDB Code 6cxs
Chain C

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Title Crystal Structure of Clostridium perfringens beta-glucuronidase bound with a novel, potent inhibitor 4-(8-(piperazin-1-yl)-1,2,3,4-tetrahydro-[1,2,3]triazino[4',5':4,5]thieno[2,3-c]isoquinolin-5-yl)morpholine
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Beta-glucuronidase
Source (MALE_ECOLI)
Sequence C:  KLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKA
KGKSALMFNLQEPYFTWPLIAADGGYAFKYENGKYDIKDV
GVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGE
TAMTINGPWAWSNIDTSKVNYGVTVLPTFKGQPSKPFVGV
LSAGINAASPNKELAVNKDKPLGAVALKSYEEELAKDPRI
AATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTV
DEALKDAQTNSS
Description


Functional site

1) chain C
residue 109-126
type prosite
sequence PIAVEALSLIYNKDLLPN
description SBP_BACTERIAL_1 Bacterial extracellular solute-binding proteins, family 1 signature. PIAvEalSLIYNkdlLpN
source prosite : PS01037


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