|
eF-site ID
|
6c3n-B |
PDB Code
|
6c3n |
Chain
|
B |
|
click to enlarge
|
|
Title
|
Crystal structure of BCL6 BTB domain in complex with compound 7CC5 |
Classification
|
TRANSCRIPTION/Inhibitor |
Compound
|
B-cell lymphoma 6 protein |
Source
|
(BCL6_HUMAN) |
|
Sequence
|
B: |
SQIQFTRHASDVLLNLNRLRSRDILTDVVIVVSREQFRAH
KTVLMACSGLFYSIFTDQLKRNLSVINLDPEINPEGFNIL
LDFMYTSRLNLRVGNIMAVMATAMYLQMEHVVDTCRKFIK
AS
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
21 |
type |
|
sequence |
N
|
description |
binding site for residue EHY A 201
|
source |
: AC1
|
|
2)
|
chain |
B |
residue |
25 |
type |
|
sequence |
L
|
description |
binding site for residue EHY A 201
|
source |
: AC1
|
|
3)
|
chain |
B |
residue |
28 |
type |
|
sequence |
R
|
description |
binding site for residue EHY B 201
|
source |
: AC2
|
|
4)
|
chain |
B |
residue |
51 |
type |
|
sequence |
M
|
description |
binding site for residue EHY B 201
|
source |
: AC2
|
|
5)
|
chain |
B |
residue |
55 |
type |
|
sequence |
G
|
description |
binding site for residue EHY B 201
|
source |
: AC2
|
|
6)
|
chain |
B |
residue |
58 |
type |
|
sequence |
Y
|
description |
binding site for residue EHY B 201
|
source |
: AC2
|
|
|
|