eF-site ID 6bu3-B
PDB Code 6bu3
Chain B

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Title CTX-M-27 Beta-Lactamase in Complex with a Non-Covalent Tetrazole Inhibitor
Classification hydrolase/hydrolase inhibitor
Compound Beta-lactamase
Source (B5LY47_ECOLX)
Sequence B:  TSAVQQKLAALEKSSGGRLGVALIDTADNTQVLYRGDERF
PMCSTSKVMAAAAVLKQSETQKQLLNQPVEIKHADLVNYN
PIAEKHVNGTMTLAELSAAALQYSDNTAMNKLIAQLGGPG
GVTAFARAIGDETFRLDRTEPTLNTAIPGDPRDTTTPRAM
AQTLRQLTLGHALGETQRAQLVTWLKGNTTGAASIRAGLP
TSWTVGDKTGSGGYGTTNDIAVIWPQGRAPLVLVTYFTQP
QQNAESRRDVLASAARIIAEGL
Description


Functional site

1) chain B
residue 222
type
sequence R
description binding site for residue 3GK A 302
source : AC2

2) chain B
residue 104
type
sequence N
description binding site for residue 3GK B 301
source : AC6

3) chain B
residue 105
type
sequence Y
description binding site for residue 3GK B 301
source : AC6

4) chain B
residue 130
type
sequence S
description binding site for residue 3GK B 301
source : AC6

5) chain B
residue 132
type
sequence N
description binding site for residue 3GK B 301
source : AC6

6) chain B
residue 167
type
sequence P
description binding site for residue 3GK B 301
source : AC6

7) chain B
residue 170
type
sequence N
description binding site for residue 3GK B 301
source : AC6

8) chain B
residue 171
type
sequence T
description binding site for residue 3GK B 301
source : AC6

9) chain B
residue 235
type
sequence T
description binding site for residue 3GK B 301
source : AC6

10) chain B
residue 236
type
sequence G
description binding site for residue 3GK B 301
source : AC6

11) chain B
residue 237
type
sequence S
description binding site for residue 3GK B 301
source : AC6

12) chain B
residue 238
type
sequence G
description binding site for residue 3GK B 301
source : AC6

13) chain B
residue 240
type
sequence G
description binding site for residue 3GK B 301
source : AC6

14) chain B
residue 104
type
sequence N
description binding site for residue 3GK B 302
source : AC7

15) chain B
residue 105
type
sequence Y
description binding site for residue 3GK B 302
source : AC7

16) chain B
residue 237
type
sequence S
description binding site for residue 3GK B 302
source : AC7

17) chain B
residue 274
type
sequence S
description binding site for residue 3GK B 302
source : AC7

18) chain B
residue 153
type
sequence R
description binding site for residue SO4 B 303
source : AC8

19) chain B
residue 108
type
sequence I
description binding site for residue SO4 B 304
source : AC9

20) chain B
residue 111
type
sequence K
description binding site for residue SO4 B 304
source : AC9

21) chain B
residue 112
type
sequence H
description binding site for residue SO4 B 304
source : AC9

22) chain B
residue 274
type
sequence S
description binding site for residue SO4 B 305
source : AD1

23) chain B
residue 275
type
sequence R
description binding site for residue SO4 B 305
source : AD1

24) chain B
residue 276
type
sequence R
description binding site for residue SO4 B 305
source : AD1

25) chain B
residue 277
type
sequence D
description binding site for residue SO4 B 305
source : AD1


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