eF-site ID 5q05-C
PDB Code 5q05
Chain C

click to enlarge
Title Human liver fructose-1,6-bisphosphatase 1 (fructose 1,6-bisphosphate 1-phosphatase, E.C.3.1.3.11) complexed with the allosteric inhibitor 1-(5-bromo-1,3-thiazol-2-yl)-3-[5-(2-methoxyethyl)-4-methylthiophen-2-yl]sulfonylurea
Classification Hydrolase/Hydrolase Inhibitor
Compound Fructose-1,6-bisphosphatase 1
Source (Q2TU34_HUMAN)
Sequence C:  DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAV
RKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEE
DKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGI
YRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMD
CGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKD
FDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVY
GGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTG
KEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS
Description


Functional site

1) chain C
residue 27
type
sequence T
description binding site for residue 95S A 401
source : AC1

2) chain C
residue 18
type
sequence M
description binding site for residue 95S C 401
source : AC3

3) chain C
residue 21
type
sequence G
description binding site for residue 95S C 401
source : AC3

4) chain C
residue 22
type
sequence R
description binding site for residue 95S C 401
source : AC3

5) chain C
residue 26
type
sequence G
description binding site for residue 95S C 401
source : AC3

6) chain C
residue 27
type
sequence T
description binding site for residue 95S C 401
source : AC3

7) chain C
residue 28
type
sequence G
description binding site for residue 95S C 401
source : AC3

8) chain C
residue 29
type
sequence E
description binding site for residue 95S C 401
source : AC3

9) chain C
residue 30
type
sequence L
description binding site for residue 95S C 401
source : AC3

10) chain C
residue 31
type
sequence T
description binding site for residue 95S C 401
source : AC3

11) chain C
residue 160
type
sequence V
description binding site for residue 95S C 401
source : AC3


Display surface

Download
Links