eF-site ID 5owk-A
PDB Code 5owk
Chain A

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Title Crystal structure of CREBBP bromodomain complexed with DSPB2A002
Classification TRANSCRIPTION
Compound CREB-binding protein
Source (CBP_HUMAN)
Sequence A:  KIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGI
PDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFN
NAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSL
Description


Functional site

1) chain A
residue 1110
type
sequence P
description binding site for residue 7MX A 1201
source : AC1

2) chain A
residue 1115
type
sequence V
description binding site for residue 7MX A 1201
source : AC1

3) chain A
residue 1120
type
sequence L
description binding site for residue 7MX A 1201
source : AC1

4) chain A
residue 1122
type
sequence I
description binding site for residue 7MX A 1201
source : AC1

5) chain A
residue 1168
type
sequence N
description binding site for residue 7MX A 1201
source : AC1

6) chain A
residue 1095
type
sequence M
description binding site for residue 7MX A 1202
source : AC2

7) chain A
residue 1099
type
sequence E
description binding site for residue 7MX A 1202
source : AC2

8) chain A
residue 1102
type
sequence Y
description binding site for residue 7MX A 1202
source : AC2

9) chain A
residue 1139
type
sequence K
description binding site for residue 7MX A 1202
source : AC2

10) chain A
residue 1151
type
sequence W
description binding site for residue 7MX A 1202
source : AC2

11) chain A
residue 1108-1167
type prosite
sequence SLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQY
QEPWQYVDDVWLMFNNAWLY
description BROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
source prosite : PS00633


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