eF-site ID 5o4s-B
PDB Code 5o4s
Chain B

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Title Crystal structure of the human BRPF1 bromodomain in complex with BZ135
Classification DNA BINDING PROTEIN
Compound Peregrin
Source (BRPF1_HUMAN)
Sequence B:  QLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDH
IKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYN
AKDTIFYRAAVRLREQGGAVLRQARRQAEKM
Description


Functional site

1) chain B
residue 639
type
sequence K
description binding site for residue 9KW A 801
source : AC1

2) chain B
residue 691
type
sequence D
description binding site for residue NO3 A 802
source : AC2

3) chain B
residue 733
type
sequence R
description binding site for residue NO3 A 802
source : AC2

4) chain B
residue 652
type
sequence I
description binding site for residue 9KW B 801
source : AC3

5) chain B
residue 658
type
sequence P
description binding site for residue 9KW B 801
source : AC3

6) chain B
residue 661
type
sequence E
description binding site for residue 9KW B 801
source : AC3

7) chain B
residue 662
type
sequence V
description binding site for residue 9KW B 801
source : AC3

8) chain B
residue 704
type
sequence C
description binding site for residue 9KW B 801
source : AC3

9) chain B
residue 707
type
sequence Y
description binding site for residue 9KW B 801
source : AC3

10) chain B
residue 708
type
sequence N
description binding site for residue 9KW B 801
source : AC3

11) chain B
residue 714
type
sequence F
description binding site for residue 9KW B 801
source : AC3


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