eF-site ID 5mwg-B
PDB Code 5mwg
Chain B

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Title Crystal structure of the human BRPF1 bromodomain in complex with BZ091
Classification DNA BINDING PROTEIN
Compound Peregrin
Source (BRPF1_HUMAN)
Sequence B:  MQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLD
HIKKPMDFFTMKQNLEAYRYLNFDDFEEDFNLIVSNCLKY
NAKDTIFYRAAVRLREQGGAVLRQARRQAEKM
Description (1)  Peregrin


Functional site

1) chain B
residue 639
type
sequence K
description binding site for residue WGX A 801
source : AC1

2) chain B
residue 652
type
sequence I
description binding site for residue WGX B 801
source : AC3

3) chain B
residue 653
type
sequence F
description binding site for residue WGX B 801
source : AC3

4) chain B
residue 657
type
sequence V
description binding site for residue WGX B 801
source : AC3

5) chain B
residue 658
type
sequence P
description binding site for residue WGX B 801
source : AC3

6) chain B
residue 661
type
sequence E
description binding site for residue WGX B 801
source : AC3

7) chain B
residue 704
type
sequence C
description binding site for residue WGX B 801
source : AC3

8) chain B
residue 707
type
sequence Y
description binding site for residue WGX B 801
source : AC3

9) chain B
residue 708
type
sequence N
description binding site for residue WGX B 801
source : AC3

10) chain B
residue 713
type
sequence I
description binding site for residue WGX B 801
source : AC3

11) chain B
residue 714
type
sequence F
description binding site for residue WGX B 801
source : AC3


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