|
eF-site ID
|
5mpk-B |
PDB Code
|
5mpk |
Chain
|
B |
|
click to enlarge
|
|
Title
|
Crystal structure of CREBBP bromodomain complexed with DK19 |
Classification
|
TRANSCRIPTION |
Compound
|
CREB-binding protein |
Source
|
(CBP_HUMAN) |
|
Sequence
|
B: |
IFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQLLGIP
DYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVWLMFNN
AWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQS
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
1110 |
type |
|
sequence |
P
|
description |
binding site for residue 0BC B 1201
|
source |
: AC2
|
|
2)
|
chain |
B |
residue |
1115 |
type |
|
sequence |
V
|
description |
binding site for residue 0BC B 1201
|
source |
: AC2
|
|
3)
|
chain |
B |
residue |
1120 |
type |
|
sequence |
L
|
description |
binding site for residue 0BC B 1201
|
source |
: AC2
|
|
4)
|
chain |
B |
residue |
1168 |
type |
|
sequence |
N
|
description |
binding site for residue 0BC B 1201
|
source |
: AC2
|
|
5)
|
chain |
B |
residue |
1173 |
type |
|
sequence |
R
|
description |
binding site for residue 0BC B 1201
|
source |
: AC2
|
|
6)
|
chain |
B |
residue |
1174 |
type |
|
sequence |
V
|
description |
binding site for residue 0BC B 1201
|
source |
: AC2
|
|
|
|