eF-site ID 5mme-AB
PDB Code 5mme
Chain A, B

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Title Crystal structure of CREBBP bromodomain complexd with US46C
Classification TRANSFERASE
Compound CREB-binding protein
Source (CBP_HUMAN)
Sequence A:  SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQ
LLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVW
LMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG
B:  SMRKKIFKPEELRQALMPTLEALYRQDPESLPFRQPVDPQ
LLGIPDYFDIVKNPMDLSTIKRKLDTGQYQEPWQYVDDVW
LMFNNAWLYNRKTSRVYKFCSKLAEVFEQEIDPVMQSLG
Description


Functional site

1) chain A
residue 1109
type
sequence L
description binding site for residue 8Q6 A 1201
source : AC1

2) chain A
residue 1110
type
sequence P
description binding site for residue 8Q6 A 1201
source : AC1

3) chain A
residue 1113
type
sequence Q
description binding site for residue 8Q6 A 1201
source : AC1

4) chain A
residue 1115
type
sequence V
description binding site for residue 8Q6 A 1201
source : AC1

5) chain A
residue 1120
type
sequence L
description binding site for residue 8Q6 A 1201
source : AC1

6) chain A
residue 1168
type
sequence N
description binding site for residue 8Q6 A 1201
source : AC1

7) chain A
residue 1173
type
sequence R
description binding site for residue 8Q6 A 1201
source : AC1

8) chain B
residue 1120
type
sequence L
description binding site for residue 8Q6 A 1201
source : AC1

9) chain B
residue 1109
type
sequence L
description binding site for residue 8Q6 B 1201
source : AC2

10) chain B
residue 1110
type
sequence P
description binding site for residue 8Q6 B 1201
source : AC2

11) chain B
residue 1120
type
sequence L
description binding site for residue 8Q6 B 1201
source : AC2

12) chain B
residue 1168
type
sequence N
description binding site for residue 8Q6 B 1201
source : AC2

13) chain B
residue 1173
type
sequence R
description binding site for residue 8Q6 B 1201
source : AC2

14) chain B
residue 1174
type
sequence V
description binding site for residue 8Q6 B 1201
source : AC2

15) chain A
residue 1108-1167
type prosite
sequence SLPFRQPVDPQLLGIPDYFDIVKNPMDLSTIKRKLDTGQY
QEPWQYVDDVWLMFNNAWLY
description BROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
source prosite : PS00633


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