eF-site ID 5mkx-B
PDB Code 5mkx
Chain B

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Title 1.68A STRUCTURE PCAF BROMODOMAIN WITH 4-chloro-2-methyl-5-(methylamino)pyridazin-3(2H)-one
Classification TRANSCRIPTION
Compound Histone acetyltransferase KAT2B
Source Homo sapiens (Human) (KAT2B_HUMAN)
Sequence B:  PDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVI
RFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNP
PESEYYKCANILEKFFFSKIKEAGLID
Description


Functional site

1) chain B
residue 729
type
sequence Y
description binding site for residue SO4 A 902
source : AC2

2) chain B
residue 780
type
sequence R
description binding site for residue SO4 A 902
source : AC2

3) chain B
residue 747
type
sequence P
description binding site for residue 82I B 901
source : AC4

4) chain B
residue 748
type
sequence F
description binding site for residue 82I B 901
source : AC4

5) chain B
residue 802
type
sequence Y
description binding site for residue 82I B 901
source : AC4

6) chain B
residue 803
type
sequence N
description binding site for residue 82I B 901
source : AC4

7) chain B
residue 809
type
sequence Y
description binding site for residue 82I B 901
source : AC4

8) chain B
residue 766
type
sequence F
description binding site for residue BU1 B 902
source : AC5


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