eF-site ID 5mkx-A
PDB Code 5mkx
Chain A

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Title 1.68A STRUCTURE PCAF BROMODOMAIN WITH 4-chloro-2-methyl-5-(methylamino)pyridazin-3(2H)-one
Classification TRANSCRIPTION
Compound Histone acetyltransferase KAT2B
Source Homo sapiens (Human) (KAT2B_HUMAN)
Sequence A:  DQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVIR
FPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNPP
ESEYYKCANILEKFFFSKIKEAGLID
Description


Functional site

1) chain A
residue 747
type
sequence P
description binding site for residue 82I A 901
source : AC1

2) chain A
residue 752
type
sequence V
description binding site for residue 82I A 901
source : AC1

3) chain A
residue 756
type
sequence E
description binding site for residue 82I A 901
source : AC1

4) chain A
residue 802
type
sequence Y
description binding site for residue 82I A 901
source : AC1

5) chain A
residue 803
type
sequence N
description binding site for residue 82I A 901
source : AC1

6) chain A
residue 809
type
sequence Y
description binding site for residue 82I A 901
source : AC1

7) chain A
residue 776
type
sequence R
description binding site for residue SO4 A 902
source : AC2

8) chain A
residue 751
type
sequence P
description binding site for residue EPE A 903
source : AC3

9) chain A
residue 754
type
sequence R
description binding site for residue EPE A 903
source : AC3

10) chain A
residue 761
type
sequence Y
description binding site for residue EPE A 903
source : AC3

11) chain A
residue 745-802
type prosite
sequence AWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVS
KKLFMADLQRVFTNCKEY
description BROMODOMAIN_1 Bromodomain signature. AwpFmepvKrteap..GYYevIrfpMdlktMserlknry..Yvskklfmadlqr.VftNCkeY
source prosite : PS00633


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