eF-site ID 5l65-b
PDB Code 5l65
Chain b

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Title Yeast 20S proteasome with mouse beta5i (1-138) and mouse beta6 (97-111; 118-133) in complex with carfilzomib
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Proteasome subunit alpha type-2
Source ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae (strain ATCC 204508 / S288c);
Sequence b:  TSIMAVTFKDGVILGADSRTTTGAYIANRVTDKLTRVHDK
IWCCRSGSAADTQAIADIVQYHLELYTSQYGTPSTETAAS
VFKELCYENKDNLTAGIIVAGYDDKNKGEVYTIPLGGSVH
KLPYAIAGSGSTFIYGYCDKNFRENMSKEETVDFIKHSLS
QAIKWDGSSGGVIRMVVLTAAGVERLIFYPDEYEQL
Description


Functional site

1) chain b
residue 45
type
sequence R
description binding site for residue CL b 202
source : AD7

2) chain b
residue 53
type
sequence Q
description binding site for residue CL b 202
source : AD7

3) chain b
residue 2
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

4) chain b
residue 3
type
sequence I
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

5) chain b
residue 17
type
sequence D
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

6) chain b
residue 20
type
sequence T
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

7) chain b
residue 21
type
sequence T
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

8) chain b
residue 22
type
sequence T
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

9) chain b
residue 33
type
sequence K
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

10) chain b
residue 45
type
sequence R
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

11) chain b
residue 46
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

12) chain b
residue 47
type
sequence G
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

13) chain b
residue 49
type
sequence A
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

14) chain b
residue 128
type
sequence G
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

15) chain b
residue 129
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

16) chain b
residue 130
type
sequence G
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

17) chain b
residue 168
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

18) chain b
residue 169
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE3

19) chain b
residue 2
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

20) chain b
residue 3
type
sequence I
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

21) chain b
residue 17
type
sequence D
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

22) chain b
residue 20
type
sequence T
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

23) chain b
residue 21
type
sequence T
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

24) chain b
residue 22
type
sequence T
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

25) chain b
residue 33
type
sequence K
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

26) chain b
residue 45
type
sequence R
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

27) chain b
residue 46
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

28) chain b
residue 47
type
sequence G
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

29) chain b
residue 49
type
sequence A
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

30) chain b
residue 128
type
sequence G
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

31) chain b
residue 129
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

32) chain b
residue 130
type
sequence G
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

33) chain b
residue 168
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

34) chain b
residue 169
type
sequence S
description binding site for Di-peptide 3BV b 201 and THR b 1
source : AE4

35) chain b
residue 1
type ACT_SITE
sequence T
description Nucleophile => ECO:0000269|PubMed:9087403
source Swiss-Prot : SWS_FT_FI1

36) chain b
residue 4-51
type prosite
sequence MAVTFKDGVILGADSRTTTGAYIANRVTDKLTRVHDKIWC
CRSGSAAD
description PROTEASOME_BETA_1 Proteasome beta-type subunits signature. LGIrVqdSVILASSkavtrgisvlkdsdd.KtrqlsphtlmsfaGeaGD
source prosite : PS00854


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