|
eF-site ID
|
5l5h-N |
PDB Code
|
5l5h |
Chain
|
N |
|
click to enlarge
|
|
Title
|
Yeast 20S proteasome with human beta5i (1-138) and human beta6 (97-111; 118-133) in complex with PR-924 |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome subunit alpha type-2 |
Source
|
null (PSB1_YEAST) |
|
Sequence
|
N: |
TSIMAVTFKDGVILGADSRTTTGAYIANRVTDKLTRVHDK
IWCCRSGSAADTQAIADIVQYHLELYTSQYGTPSTETAAS
VFKELCYENKDNLTAGIIVAGYDDKNKGEVYTIPLGGSVH
KLPYAIAGSGSTFIYGYCDKNFRENMSKEETVDFIKHSLS
QAIKWDGSSGGVIRMVVLTAAGVERLIFYPDEYEQL
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
N |
residue |
163 |
type |
|
sequence |
I
|
description |
binding site for residue MG N 201
|
source |
: AC9
|
|
2)
|
chain |
N |
residue |
166 |
type |
|
sequence |
D
|
description |
binding site for residue MG N 201
|
source |
: AC9
|
|
3)
|
chain |
N |
residue |
169 |
type |
|
sequence |
S
|
description |
binding site for residue MG N 201
|
source |
: AC9
|
|
4)
|
chain |
N |
residue |
51 |
type |
|
sequence |
D
|
description |
binding site for residue MG N 202
|
source |
: AD1
|
|
5)
|
chain |
N |
residue |
1 |
type |
ACT_SITE |
sequence |
T
|
description |
Nucleophile => ECO:0000269|PubMed:9087403
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
|
|