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eF-site ID
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5l5e-X |
PDB Code
|
5l5e |
Chain
|
X |
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click to enlarge
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Title
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Yeast 20S proteasome with human beta5i (1-138) and human beta6 (97-111; 118-133) in complex with carfilzomib |
Classification
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HYDROLASE/HYDROLASE INHIBITOR |
Compound
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Proteasome subunit alpha type-2 |
Source
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Saccharomyces cerevisiae (strain ATCC 204508 / S288c) (Baker's yeast) (PSB1_YEAST) |
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Sequence
|
X: |
MDIILGIRVQDSVILASSKAVTRGISVLKDSDDKTRQLSP
HTLMSFAGEAGDTVQFAEYIQANIQLYSIREDYELSPQAV
SSFVRQELAKSIRSRRPYQVNVLIGGYDKKKNKPELYQID
YLGTKVELPYGAHGYSGFYTFSLLDHHYRPDMTTEEGLDL
LKLCVQELEKRMPMDFKGVIVKIVDKDGIRQVDDF
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Description
|
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Functional site
|
|
1)
|
chain |
X |
residue |
76 |
type |
MOD_RES |
sequence |
S
|
description |
Phosphoserine => ECO:0007744|PubMed:18407956
|
source |
Swiss-Prot : SWS_FT_FI2
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