eF-site ID 5l5e-Y
PDB Code 5l5e
Chain Y

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Title Yeast 20S proteasome with human beta5i (1-138) and human beta6 (97-111; 118-133) in complex with carfilzomib
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Proteasome subunit alpha type-2
Source Saccharomyces cerevisiae (strain ATCC 204508 / S288c) (Baker's yeast) (PSB1_YEAST)
Sequence Y:  TTTLAFKFQHGVIAAVDSRASAGSYISALRVNKVIEINPY
LLGTMSGCAADCQYWERLLAKECRLYYLRNGERISVSAAS
KLLSNMMCQYRGMGLSMGSMICGWDKKGPGLYYVDEHGTR
LSGNMFSTGSGNTYAYGVLDSNYKWDLSVEDALYLGKRSI
LAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKVK
EEEGSFNNVIG
Description


Functional site

1) chain Y
residue 19
type
sequence R
description binding site for residue MG I 302
source : AC6

2) chain Y
residue 164
type
sequence A
description binding site for residue MG I 302
source : AC6

3) chain Y
residue 167
type
sequence D
description binding site for residue MG I 302
source : AC6

4) chain Y
residue 168
type
sequence A
description binding site for residue MG I 302
source : AC6

5) chain Y
residue 170
type
sequence S
description binding site for residue MG I 302
source : AC6

6) chain Y
residue 2
type
sequence T
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

7) chain Y
residue 3
type
sequence T
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

8) chain Y
residue 17
type
sequence D
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

9) chain Y
residue 19
type
sequence R
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

10) chain Y
residue 20
type
sequence A
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

11) chain Y
residue 27
type
sequence S
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

12) chain Y
residue 33
type
sequence K
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

13) chain Y
residue 45
type
sequence M
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

14) chain Y
residue 47
type
sequence G
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

15) chain Y
residue 49
type
sequence A
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

16) chain Y
residue 129
type
sequence G
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

17) chain Y
residue 130
type
sequence S
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

18) chain Y
residue 131
type
sequence G
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

19) chain Y
residue 169
type
sequence Y
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

20) chain Y
residue 170
type
sequence S
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE1

21) chain Y
residue 2
type
sequence T
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

22) chain Y
residue 3
type
sequence T
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

23) chain Y
residue 17
type
sequence D
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

24) chain Y
residue 19
type
sequence R
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

25) chain Y
residue 20
type
sequence A
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

26) chain Y
residue 27
type
sequence S
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

27) chain Y
residue 33
type
sequence K
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

28) chain Y
residue 45
type
sequence M
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

29) chain Y
residue 47
type
sequence G
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

30) chain Y
residue 49
type
sequence A
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

31) chain Y
residue 129
type
sequence G
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

32) chain Y
residue 130
type
sequence S
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

33) chain Y
residue 131
type
sequence G
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

34) chain Y
residue 169
type
sequence Y
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2

35) chain Y
residue 170
type
sequence S
description binding site for Di-peptide 3BV Y 301 and THR Y 1
source : AE2


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