|
eF-site ID
|
5l5e-C |
PDB Code
|
5l5e |
Chain
|
C |
|
click to enlarge
|
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Title
|
Yeast 20S proteasome with human beta5i (1-138) and human beta6 (97-111; 118-133) in complex with carfilzomib |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome subunit alpha type-2 |
Source
|
null (PSB1_YEAST) |
|
Sequence
|
C: |
GYDRALSIFSPDGHIFQVEYALEAVKRGTCAVGVKGKNCV
VLGCERRSTLKLQDTRITPSKVSKIDSHVVLSFSGLNADS
RILIEKARVEAQSHRLTLEDPVTVEYLTRYVAGVQQRYTQ
SGGVRPFGVSTLIAGFDPRDDEPKLYQTEPSGIYSSWSAQ
TIGRNSKTVREFLEKNYDRKEPPATVEECVKLTVRSLLEV
VQTGAKNIEITVVKPDSDIVALSSEEINQYVTQIEQEKQE
|
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Description
|
|
Functional site
|
|
1)
|
chain |
C |
residue |
2-24 |
type |
prosite |
sequence |
YDRALSIFSPDGHIFQVEYALEA
|
description |
PROTEASOME_ALPHA_1 Proteasome alpha-type subunits signature. YdralSiFSPdGHifQVEYAleA
|
source |
prosite : PS00388
|
|
2)
|
chain |
C |
residue |
32-79 |
type |
prosite |
sequence |
VGVKGKNCVVLGCERRSTLKLQDTRITPSKVSKIDSHVVL
SFSGLNAD
|
description |
PROTEASOME_BETA_1 Proteasome beta-type subunits signature. VGVkFnnGVVIAADtrstqgpivadknca.KlhrispkiwcagaGtaAD
|
source |
prosite : PS00854
|
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|
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