eF-site ID 5hbh-B
PDB Code 5hbh
Chain B

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Title CDK8-CYCC IN COMPLEX WITH 5-{5-Chloro-4-[1-(2-methoxy-ethyl)-1,8-diaza-spiro[4.5]dec-8-yl]-pyridin-3-yl}-1-methyl-1,3-dihydro-benzo[c]isothiazole 2,2-dioxide
Classification TRANSFERASE
Compound Cyclin-dependent kinase 8
Source Homo sapiens (Human) (CCNC_HUMAN)
Sequence B:  DDDDKAMAGNFWQSSHYLQWILDKQDLLKERQKDLKFLSE
EEYWKLQIFFTNVIQALGEHLKLRQQVIATATVYFKRFYA
RYSLKSIDPVLMAPTCVFLASKVEEFGVVSNTRLIAAATS
VLKTRFSYAFPKEFPYRMNHILECEFYLLELMDCCLIVYH
PYRPLLQYVQDMGQEDMLLPLAWRIVNDTYRTDLCLLYPP
FMIALACLHVACVVQQKDARQWFAELSVDMEKILEIIRVI
LKLYEQWKNFDERKEMATILSKMPKPKPPP
Description


Functional site

1) chain B
residue 248
type
sequence K
description binding site for residue FMT A 403
source : AC3

2) chain B
residue 203
type
sequence H
description binding site for residue FMT B 301
source : AC4

3) chain B
residue 211
type
sequence K
description binding site for residue FMT B 301
source : AC4

4) chain B
residue 213
type
sequence A
description binding site for residue FMT B 301
source : AC4

5) chain B
residue 0
type
sequence A
description binding site for residue FMT B 302
source : AC5

6) chain B
residue 152
type
sequence V
description binding site for residue FMT B 302
source : AC5

7) chain B
residue 157
type
sequence R
description binding site for residue FMT B 302
source : AC5


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