eF-site ID 5fe9-AB
PDB Code 5fe9
Chain A, B

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Title Crystal structure of human PCAF bromodomain in complex with compound SL1122 (compound 13)
Classification SIGNALING PROTEIN
Compound Histone acetyltransferase KAT2B
Source Homo sapiens (Human) (KAT2B_HUMAN)
Sequence A:  RDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYE
VIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEY
NPPESEYYKCANILEKFFFSKIKEAGLID
B:  RDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYE
VIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEY
NPPESEYYKCANILEKFFFSKIKEAGLID
Description


Functional site

1) chain A
residue 747
type
sequence P
description binding site for residue 5WS A 901
source : AC1

2) chain A
residue 750
type
sequence E
description binding site for residue 5WS A 901
source : AC1

3) chain A
residue 751
type
sequence P
description binding site for residue 5WS A 901
source : AC1

4) chain A
residue 753
type
sequence K
description binding site for residue 5WS A 901
source : AC1

5) chain A
residue 756
type
sequence E
description binding site for residue 5WS A 901
source : AC1

6) chain A
residue 757
type
sequence A
description binding site for residue 5WS A 901
source : AC1

7) chain A
residue 803
type
sequence N
description binding site for residue 5WS A 901
source : AC1

8) chain A
residue 780
type
sequence R
description binding site for residue EDO A 902
source : AC2

9) chain B
residue 776
type
sequence R
description binding site for residue EDO A 902
source : AC2

10) chain B
residue 781
type
sequence Y
description binding site for residue EDO A 902
source : AC2

11) chain B
residue 747
type
sequence P
description binding site for residue 5WS B 901
source : AC3

12) chain B
residue 750
type
sequence E
description binding site for residue 5WS B 901
source : AC3

13) chain B
residue 751
type
sequence P
description binding site for residue 5WS B 901
source : AC3

14) chain B
residue 752
type
sequence V
description binding site for residue 5WS B 901
source : AC3

15) chain B
residue 753
type
sequence K
description binding site for residue 5WS B 901
source : AC3

16) chain B
residue 756
type
sequence E
description binding site for residue 5WS B 901
source : AC3

17) chain B
residue 803
type
sequence N
description binding site for residue 5WS B 901
source : AC3

18) chain B
residue 809
type
sequence Y
description binding site for residue 5WS B 901
source : AC3

19) chain A
residue 745-802
type prosite
sequence AWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVS
KKLFMADLQRVFTNCKEY
description BROMODOMAIN_1 Bromodomain signature. AwpFmepvKrteap..GYYevIrfpMdlktMserlknry..Yvskklfmadlqr.VftNCkeY
source prosite : PS00633


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