eF-site ID 5fe9-A
PDB Code 5fe9
Chain A

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Title Crystal structure of human PCAF bromodomain in complex with compound SL1122 (compound 13)
Classification SIGNALING PROTEIN
Compound Histone acetyltransferase KAT2B
Source Homo sapiens (Human) (KAT2B_HUMAN)
Sequence A:  RDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYE
VIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEY
NPPESEYYKCANILEKFFFSKIKEAGLID
Description


Functional site

1) chain A
residue 747
type
sequence P
description binding site for residue 5WS A 901
source : AC1

2) chain A
residue 750
type
sequence E
description binding site for residue 5WS A 901
source : AC1

3) chain A
residue 751
type
sequence P
description binding site for residue 5WS A 901
source : AC1

4) chain A
residue 753
type
sequence K
description binding site for residue 5WS A 901
source : AC1

5) chain A
residue 756
type
sequence E
description binding site for residue 5WS A 901
source : AC1

6) chain A
residue 757
type
sequence A
description binding site for residue 5WS A 901
source : AC1

7) chain A
residue 803
type
sequence N
description binding site for residue 5WS A 901
source : AC1

8) chain A
residue 780
type
sequence R
description binding site for residue EDO A 902
source : AC2

9) chain A
residue 745-802
type prosite
sequence AWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVS
KKLFMADLQRVFTNCKEY
description BROMODOMAIN_1 Bromodomain signature. AwpFmepvKrteap..GYYevIrfpMdlktMserlknry..Yvskklfmadlqr.VftNCkeY
source prosite : PS00633


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