eF-site ID 5fe9-B
PDB Code 5fe9
Chain B

click to enlarge
Title Crystal structure of human PCAF bromodomain in complex with compound SL1122 (compound 13)
Classification SIGNALING PROTEIN
Compound Histone acetyltransferase KAT2B
Source Homo sapiens (Human) (KAT2B_HUMAN)
Sequence B:  RDPDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYE
VIRFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEY
NPPESEYYKCANILEKFFFSKIKEAGLID
Description


Functional site

1) chain B
residue 776
type
sequence R
description binding site for residue EDO A 902
source : AC2

2) chain B
residue 781
type
sequence Y
description binding site for residue EDO A 902
source : AC2

3) chain B
residue 747
type
sequence P
description binding site for residue 5WS B 901
source : AC3

4) chain B
residue 750
type
sequence E
description binding site for residue 5WS B 901
source : AC3

5) chain B
residue 751
type
sequence P
description binding site for residue 5WS B 901
source : AC3

6) chain B
residue 752
type
sequence V
description binding site for residue 5WS B 901
source : AC3

7) chain B
residue 753
type
sequence K
description binding site for residue 5WS B 901
source : AC3

8) chain B
residue 756
type
sequence E
description binding site for residue 5WS B 901
source : AC3

9) chain B
residue 803
type
sequence N
description binding site for residue 5WS B 901
source : AC3

10) chain B
residue 809
type
sequence Y
description binding site for residue 5WS B 901
source : AC3


Display surface

Download
Links