eF-site ID 5fe2-B
PDB Code 5fe2
Chain B

click to enlarge
Title Crystal structure of human PCAF bromodomain in complex with fragment BR013 (fragment 3)
Classification SIGNALING PROTEIN
Compound Histone acetyltransferase KAT2B
Source Homo sapiens (Human) (KAT2B_HUMAN)
Sequence B:  PDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVI
RFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNP
PESEYYKCANILEKFFFSKIKEAGLID
Description


Functional site

1) chain B
residue 747
type
sequence P
description binding site for residue 5WV B 901
source : AC3

2) chain B
residue 756
type
sequence E
description binding site for residue 5WV B 901
source : AC3

3) chain B
residue 757
type
sequence A
description binding site for residue 5WV B 901
source : AC3

4) chain B
residue 803
type
sequence N
description binding site for residue 5WV B 901
source : AC3

5) chain B
residue 809
type
sequence Y
description binding site for residue 5WV B 901
source : AC3

6) chain B
residue 743
type
sequence Q
description binding site for residue EDO B 902
source : AC4

7) chain B
residue 744
type
sequence S
description binding site for residue EDO B 902
source : AC4

8) chain B
residue 815
type
sequence I
description binding site for residue EDO B 902
source : AC4

9) chain B
residue 754
type
sequence R
description binding site for residue EDO B 903
source : AC5

10) chain B
residue 727
type
sequence Q
description binding site for residue EDO B 904
source : AC6


Display surface

Download
Links