eF-site ID 5fe2-A
PDB Code 5fe2
Chain A

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Title Crystal structure of human PCAF bromodomain in complex with fragment BR013 (fragment 3)
Classification SIGNALING PROTEIN
Compound Histone acetyltransferase KAT2B
Source Homo sapiens (Human) (KAT2B_HUMAN)
Sequence A:  PDQLYSTLKSILQQVKSHQSAWPFMEPVKRTEAPGYYEVI
RFPMDLKTMSERLKNRYYVSKKLFMADLQRVFTNCKEYNP
PESEYYKCANILEKFFFSKIKEAGLID
Description


Functional site

1) chain A
residue 747
type
sequence P
description binding site for residue 5WV A 901
source : AC1

2) chain A
residue 748
type
sequence F
description binding site for residue 5WV A 901
source : AC1

3) chain A
residue 756
type
sequence E
description binding site for residue 5WV A 901
source : AC1

4) chain A
residue 803
type
sequence N
description binding site for residue 5WV A 901
source : AC1

5) chain A
residue 733
type
sequence K
description binding site for residue EDO A 902
source : AC2

6) chain A
residue 737
type
sequence Q
description binding site for residue EDO A 902
source : AC2

7) chain A
residue 740
type
sequence K
description binding site for residue EDO A 902
source : AC2

8) chain A
residue 774
type
sequence S
description binding site for residue EDO A 902
source : AC2

9) chain A
residue 777
type
sequence L
description binding site for residue EDO A 902
source : AC2

10) chain A
residue 808
type
sequence E
description binding site for residue EDO B 904
source : AC6

11) chain A
residue 745-802
type prosite
sequence AWPFMEPVKRTEAPGYYEVIRFPMDLKTMSERLKNRYYVS
KKLFMADLQRVFTNCKEY
description BROMODOMAIN_1 Bromodomain signature. AwpFmepvKrteap..GYYevIrfpMdlktMserlknry..Yvskklfmadlqr.VftNCkeY
source prosite : PS00633


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