eF-site ID 5dkh-B
PDB Code 5dkh
Chain B

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Title Crystal structure of the bromodomain of human BRM (SMARCA2) in complex with a hydroxyphenyl propenone inhibitor 17
Classification TRANSCRIPTION
Compound Probable global transcription activator SNF2L2
Source Homo sapiens (Human) (SMCA2_HUMAN)
Sequence B:  PKLTKQMNAIIDTVINYKDSSGRQLSEVFIQLPSRKELPE
YYELIRKPVDFKKIKERIRNHKYRSLGDLEKDVMLLCHNA
QTFNLEGSQIYEDSIVLQSVFKSARQKIAK
Description


Functional site

1) chain B
residue 1441
type
sequence H
description binding site for residue ZN B 1501
source : AC4

2) chain B
residue 1458
type
sequence H
description binding site for residue ZN B 1501
source : AC4

3) chain B
residue 1441
type
sequence H
description binding site for residue ZN B 1502
source : AC5

4) chain B
residue 1458
type
sequence H
description binding site for residue ZN B 1502
source : AC5

5) chain B
residue 1467
type
sequence G
description binding site for residue EDO B 1503
source : AC6

6) chain B
residue 1472
type
sequence E
description binding site for residue EDO B 1503
source : AC6

7) chain B
residue 1417
type
sequence E
description binding site for residue EDO B 1504
source : AC7

8) chain B
residue 1408
type
sequence V
description binding site for residue 5C0 B 1505
source : AC8

9) chain B
residue 1409
type
sequence F
description binding site for residue 5C0 B 1505
source : AC8

10) chain B
residue 1412
type
sequence L
description binding site for residue 5C0 B 1505
source : AC8

11) chain B
residue 1421
type
sequence Y
description binding site for residue 5C0 B 1505
source : AC8

12) chain B
residue 1429
type
sequence V
description binding site for residue 5C0 B 1505
source : AC8

13) chain B
residue 1460
type
sequence A
description binding site for residue 5C0 B 1505
source : AC8

14) chain B
residue 1464
type
sequence N
description binding site for residue 5C0 B 1505
source : AC8

15) chain B
residue 1470
type
sequence I
description binding site for residue 5C0 B 1505
source : AC8


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