eF-site ID 5cz8-P
PDB Code 5cz8
Chain P

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Title Yeast 20S proteasome beta5-L(-49)S-K33A mutant in complex with Carfilzomib
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Proteasome subunit alpha type-2
Source ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae (strain ATCC 204508 / S288c);
Sequence P:  GSRRYDSRTTIFSPEGRLYQVEYALESISHAGTAIGIMAS
DGIVLAAERKVTSTLLEQDTSTEKLYKLNDKIAVAVAGLT
ADAEILINTARIHAQNYLKTYNEDIPVEILVRRLSDIKQG
YTQHGGLRPFGVSFIYAGYDDRYGYQLYTSNPSGNYTGWK
AISVGANTSAAQTLLQMDYKDDMKVDDAIELALKTLSKTT
DSSALTYDRLEFATIRKGANDGEVYQKIFKPQEIKDILVK
TGIT
Description


Functional site

1) chain P
residue 99
type ACT_SITE
sequence K
description Nucleophile => ECO:0000269|PubMed:9087403
source Swiss-Prot : SWS_FT_FI1

2) chain P
residue 198
type ACT_SITE
sequence K
description Nucleophile => ECO:0000269|PubMed:9087403
source Swiss-Prot : SWS_FT_FI1

3) chain P
residue 230
type ACT_SITE
sequence K
description Nucleophile => ECO:0000269|PubMed:9087403
source Swiss-Prot : SWS_FT_FI1


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