eF-site ID 5cen-A
PDB Code 5cen
Chain A

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Title Crystal structure of DLK (kinase domain)
Classification TRANSFERASE
Compound Mitogen-activated protein kinase kinase kinase 12
Source Homo sapiens (Human) (M3K12_HUMAN)
Sequence A:  LWEVPFEEILDLQWVGSGAQGAVFLGRFHGEEVAVKKVRD
LKETDIKHLRKLKHPNIITFKGVCTQAPCYCILMEFCAQG
QLYEVLRAGRPVTPSLLVDWSMGIAGGMNYLHLHKIIHRD
LKSPNMLITYDDVVKISDFGTSKELSDKSTKMSFAGTVAW
MAPEVIRNEPVSEKVDIWSFGVVLWELLTGEIPYKDVDSS
AIIWGVGSNSLHLPVPSSCPDGFKILLRQCWNSKPRNRPS
FRQILLHLDIASADVLSTPQETYFKSQAEWREEVKLHFEK
I
Description


Functional site

1) chain A
residue 232-244
type prosite
sequence IIHRDLKSPNMLI
description PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. IiHrDLKspNMLI
source prosite : PS00108

2) chain A
residue 236
type ACT_SITE
sequence D
description Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00159, ECO:0000255|PROSITE-ProRule:PRU10027
source Swiss-Prot : SWS_FT_FI1

3) chain A
residue 131
type BINDING
sequence V
description BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
source Swiss-Prot : SWS_FT_FI2

4) chain A
residue 152
type BINDING
sequence K
description BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
source Swiss-Prot : SWS_FT_FI2


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