|
eF-site ID
|
5bnj-B |
PDB Code
|
5bnj |
Chain
|
B |
|
click to enlarge
|
|
Title
|
CDK8/CYCC IN COMPLEX WITH 8-{3-Chloro-5-[4-(1-methyl-1H-pyrazol-4-yl)-phenyl]-pyridin- 4-yl}-2,8-diaza-spiro[4.5]decan-1-one |
Classification
|
TRANSFERASE |
Compound
|
Cyclin-dependent kinase 8 |
Source
|
Homo sapiens (Human) (CCNC_HUMAN) |
|
Sequence
|
B: |
KAMAGNFWQSSHYLQWILDKQDLLKERQKDLKFLSEEEYW
KLQIFFTNVIQALGEHLKLRQQVIATATVYFKRFYARYSL
KSIDPVLMAPTCVFLASKVEEFGVVSNTRLIAAATSVLKT
RFSYAFPKEFPYRMNHILECEFYLLELMDCCLIVYHPYRP
LLQYVQDMGQEDMLLPLAWRIVNDTYRTDLCLLYPPFMIA
LACLHVACVVQQKDARQWFAELSVDMEKILEIIRVILKLY
EQWKNFDERKEMATILSKMPKPKPPP
|
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Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
144 |
type |
|
sequence |
E
|
description |
binding site for residue FMT B 301
|
source |
: AC2
|
|
2)
|
chain |
B |
residue |
147 |
type |
|
sequence |
D
|
description |
binding site for residue FMT B 302
|
source |
: AC3
|
|
|
|