|
eF-site ID
|
5ame-A |
PDB Code
|
5ame |
Chain
|
A |
|
click to enlarge
|
|
Title
|
Crystal structure of the bromodomain of human surface epitope engineered BRD1A in complex with 3D Consortium fragment 4-acetyl- piperazin-2-one (SGC - Diamond I04-1 fragment screening) |
Classification
|
TRANSCRIPTION |
Compound
|
BROMODOMAIN-CONTAINING PROTEIN 1 |
Source
|
(BRD1_HUMAN) |
|
Sequence
|
A: |
SMEQVAMELRLTELTRLLRSVLDQLQDKDPARIFAQPVSL
KEVPDYLDHIKHPMDFATMRKRLEAQGYKNLHEFEEDFDL
IIDNCMKYNARDTVFYRAAVRLRDQGGVVLRQARREVDSI
GLE
|
|
Description
|
(1) |
BROMODOMAIN-CONTAINING PROTEIN 1
|
|
Functional site
|
|
1)
|
chain |
A |
residue |
108 |
type |
|
sequence |
K
|
description |
BINDING SITE FOR RESIDUE NA B 1146
|
source |
: AC2
|
|
2)
|
chain |
A |
residue |
62 |
type |
CROSSLNK |
sequence |
K
|
description |
Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
3)
|
chain |
A |
residue |
52-109 |
type |
prosite |
sequence |
ARIFAQPVSLKEVPDYLDHIKHPMDFATMRKRLEAQGYKN
LHEFEEDFDLIIDNCMKY
|
description |
BROMODOMAIN_1 Bromodomain signature. AriFaqpvSlkevp..DYLdhIkhpMdfatMrkrleaqg..Yknlhefeedfdl.IidNCmkY
|
source |
prosite : PS00633
|
|
|
|