eF-site ID 5ame-A
PDB Code 5ame
Chain A

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Title Crystal structure of the bromodomain of human surface epitope engineered BRD1A in complex with 3D Consortium fragment 4-acetyl- piperazin-2-one (SGC - Diamond I04-1 fragment screening)
Classification TRANSCRIPTION
Compound BROMODOMAIN-CONTAINING PROTEIN 1
Source (BRD1_HUMAN)
Sequence A:  SMEQVAMELRLTELTRLLRSVLDQLQDKDPARIFAQPVSL
KEVPDYLDHIKHPMDFATMRKRLEAQGYKNLHEFEEDFDL
IIDNCMKYNARDTVFYRAAVRLRDQGGVVLRQARREVDSI
GLE
Description (1)  BROMODOMAIN-CONTAINING PROTEIN 1


Functional site

1) chain A
residue 108
type
sequence K
description BINDING SITE FOR RESIDUE NA B 1146
source : AC2

2) chain A
residue 62
type CROSSLNK
sequence K
description Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
source Swiss-Prot : SWS_FT_FI1

3) chain A
residue 52-109
type prosite
sequence ARIFAQPVSLKEVPDYLDHIKHPMDFATMRKRLEAQGYKN
LHEFEEDFDLIIDNCMKY
description BROMODOMAIN_1 Bromodomain signature. AriFaqpvSlkevp..DYLdhIkhpMdfatMrkrleaqg..Yknlhefeedfdl.IidNCmkY
source prosite : PS00633


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