eF-site ID 4tyl-A
PDB Code 4tyl
Chain A

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Title Fragment-Based Screening of the Bromodomain of ATAD2
Classification Hydrolase/Hydrolase inhibitor
Compound ATPase family AAA domain-containing protein 2
Source (ATAD2_HUMAN)
Sequence A:  SMQEEDTFRELRIFLRNVTHRLAIDKRFRVFTKPVDPDEV
PDYVTVIKQPMDLSSVISKIDLHKYLTVKDYLRDIDLICS
NALEYNPDRDPGDRLIRHRACALRDTAYAIIKEELDEDFE
QLCEEIQESR
Description


Functional site

1) chain A
residue 987
type
sequence R
description binding site for residue SO4 A 1201
source : AC1

2) chain A
residue 990
type
sequence R
description binding site for residue SO4 A 1201
source : AC1

3) chain A
residue 994
type
sequence R
description binding site for residue SO4 A 1201
source : AC1

4) chain A
residue 1067
type
sequence R
description binding site for residue SO4 A 1201
source : AC1

5) chain A
residue 1072
type
sequence R
description binding site for residue SO4 A 1201
source : AC1

6) chain A
residue 1077
type
sequence R
description binding site for residue CL A 1202
source : AC2

7) chain A
residue 1008
type
sequence V
description binding site for residue 39O A 1203
source : AC3

8) chain A
residue 1013
type
sequence V
description binding site for residue 39O A 1203
source : AC3

9) chain A
residue 1063
type
sequence Y
description binding site for residue 39O A 1203
source : AC3

10) chain A
residue 1064
type
sequence N
description binding site for residue 39O A 1203
source : AC3

11) chain A
residue 1074
type
sequence I
description binding site for residue 39O A 1203
source : AC3


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