eF-site ID 4qwu-Y
PDB Code 4qwu
Chain Y

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Title yCP beta5-C52F mutant in complex with bortezomib
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Proteasome subunit alpha type-2
Source ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae;
Sequence Y:  TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPF
LLGTMAGGAADFQFWETWLGSQCRLHELREKERISVAAAS
KILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGT
RLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRS
ILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKV
KEEEGSFNNVIG
Description


Functional site

1) chain Y
residue 1
type
sequence T
description BINDING SITE FOR RESIDUE BO2 Y 301
source : BC4

2) chain Y
residue 20
type
sequence A
description BINDING SITE FOR RESIDUE BO2 Y 301
source : BC4

3) chain Y
residue 21
type
sequence T
description BINDING SITE FOR RESIDUE BO2 Y 301
source : BC4

4) chain Y
residue 45
type
sequence M
description BINDING SITE FOR RESIDUE BO2 Y 301
source : BC4

5) chain Y
residue 47
type
sequence G
description BINDING SITE FOR RESIDUE BO2 Y 301
source : BC4

6) chain Y
residue 48
type
sequence G
description BINDING SITE FOR RESIDUE BO2 Y 301
source : BC4

7) chain Y
residue 49
type
sequence A
description BINDING SITE FOR RESIDUE BO2 Y 301
source : BC4

8) chain Y
residue 170
type
sequence Y
description BINDING SITE FOR RESIDUE BO2 Y 301
source : BC4

9) chain Y
residue 165
type
sequence A
description BINDING SITE FOR RESIDUE MG Y 302
source : BC5

10) chain Y
residue 168
type
sequence D
description BINDING SITE FOR RESIDUE MG Y 302
source : BC5

11) chain Y
residue 169
type
sequence A
description BINDING SITE FOR RESIDUE MG Y 302
source : BC5

12) chain Y
residue 171
type
sequence S
description BINDING SITE FOR RESIDUE MG Y 302
source : BC5

13) chain Y
residue 49
type BINDING
sequence A
description
source Swiss-Prot : SWS_FT_FI2


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