|
eF-site ID
|
4qwu-J |
PDB Code
|
4qwu |
Chain
|
J |
|
click to enlarge
|
|
Title
|
yCP beta5-C52F mutant in complex with bortezomib |
Classification
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HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome subunit alpha type-2 |
Source
|
ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
J: |
MDIILGIRVQDSVILASSKAVTRGISVLKDSDDKTRQLSP
HTLMSFAGEAGDTVQFAEYIQANIQLYSIREDYELSPQAV
SSFVRQELAKSIRSRRPYQVNVLIGGYDKKKNKPELYQID
YLGTKVELPYGAHGYSGFYTFSLLDHHYRPDMTTEEGLDL
LKLCVQELEKRMPMDFKGVIVKIVDKDGIRQVDDF
|
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Description
|
|
Functional site
|
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1)
|
chain |
J |
residue |
118 |
type |
|
sequence |
Q
|
description |
BINDING SITE FOR RESIDUE MG J 201
|
source |
: AC4
|
|
2)
|
chain |
J |
residue |
120 |
type |
|
sequence |
D
|
description |
BINDING SITE FOR RESIDUE MG J 201
|
source |
: AC4
|
|
3)
|
chain |
J |
residue |
124 |
type |
|
sequence |
T
|
description |
BINDING SITE FOR RESIDUE MG J 201
|
source |
: AC4
|
|
4)
|
chain |
J |
residue |
5-52 |
type |
prosite |
sequence |
LGIRVQDSVILASSKAVTRGISVLKDSDDKTRQLSPHTLM
SFAGEAGD
|
description |
PROTEASOME_BETA_1 Proteasome beta-type subunits signature. VAMtGkdCVAIACDlrlgsqslgvsnkfe.Kifhyghvflgit.GlaTD
|
source |
prosite : PS00854
|
|
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