|
eF-site ID
|
4qwr-U |
PDB Code
|
4qwr |
Chain
|
U |
|
click to enlarge
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|
Title
|
yCP beta5-C52F mutant in complex with carfilzomib |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome subunit alpha type-2 |
Source
|
ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
U: |
GYDRHITIFSPEGRLYQVEYAFKATNQTNINSLAVRGKDC
TVVISQKKVPDKLLDPTTVSYIFCISRTIGMVVNGPIPDA
RNAALRAKAEAAEFRYKYGYDMPCDVLAKRMANLSQIYTQ
RAYMRPLGVILTFVSVDEELGPSIYKTDPAGYYVGYKATA
TGPKQQEITTNLENHFKKSKIDHINEESWEKVVEFAITHM
IDALGTEFSKNDLEVGVATKDKFFTLSAENIEERLVAIAE
Q
|
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Description
|
|
Functional site
|
|
1)
|
chain |
U |
residue |
111 |
type |
|
sequence |
R
|
description |
BINDING SITE FOR RESIDUE CL U 301
|
source |
: BC3
|
|
2)
|
chain |
U |
residue |
114 |
type |
|
sequence |
N
|
description |
BINDING SITE FOR RESIDUE CL U 301
|
source |
: BC3
|
|
3)
|
chain |
U |
residue |
223 |
type |
CROSSLNK |
sequence |
K
|
description |
Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0007744|PubMed:22106047
|
source |
Swiss-Prot : SWS_FT_FI3
|
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