|
eF-site ID
|
4qwl-X |
PDB Code
|
4qwl |
Chain
|
X |
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click to enlarge
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Title
|
yCP beta5-A50V mutant in complex with carfilzomib |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
Proteasome subunit alpha type-2 |
Source
|
ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
X: |
MDIILGIRVQDSVILASSKAVTRGISVLKDSDDKTRQLSP
HTLMSFAGEAGDTVQFAEYIQANIQLYSIREDYELSPQAV
SSFVRQELAKSIRSRRPYQVNVLIGGYDKKKNKPELYQID
YLGTKVELPYGAHGYSGFYTFSLLDHHYRPDMTTEEGLDL
LKLCVQELEKRMPMDFKGVIVKIVDKDGIRQVDDF
|
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Description
|
|
Functional site
|
|
1)
|
chain |
X |
residue |
23 |
type |
|
sequence |
R
|
description |
BINDING SITE FOR RESIDUE MES X 201
|
source |
: BC6
|
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