eF-site ID 4qwl-Y
PDB Code 4qwl
Chain Y

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Title yCP beta5-A50V mutant in complex with carfilzomib
Classification HYDROLASE/HYDROLASE INHIBITOR
Compound Proteasome subunit alpha type-2
Source ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae;
Sequence Y:  TTTLAFRFQGGIIVAVDSRATAGNWVASQTVKKVIEINPF
LLGTMAGGAVDCQFWETWLGSQCRLHELREKERISVAAAS
KILSNLVYQYKGAGLSMGTMICGYTRKEGPTIYYVDSDGT
RLKGDIFCVGSGQTFAYGVLDSNYKWDLSVEDALYLGKRS
ILAAAHRDAYSGGSVNLYHVTEDGWIYHGNHDVGELFWKV
KEEEGSFNNVIG
Description


Functional site

1) chain Y
residue 1
type
sequence T
description BINDING SITE FOR RESIDUE MES X 201
source : BC6

2) chain Y
residue 47
type
sequence G
description BINDING SITE FOR RESIDUE MES X 201
source : BC6

3) chain Y
residue 97
type
sequence M
description BINDING SITE FOR RESIDUE MES X 201
source : BC6

4) chain Y
residue 117
type
sequence S
description BINDING SITE FOR RESIDUE MES X 201
source : BC6

5) chain Y
residue 130
type
sequence G
description BINDING SITE FOR RESIDUE MES X 201
source : BC6

6) chain Y
residue 131
type
sequence S
description BINDING SITE FOR RESIDUE MES X 201
source : BC6

7) chain Y
residue 1
type
sequence T
description BINDING SITE FOR RESIDUE 3BV Y 301
source : BC7

8) chain Y
residue 19
type
sequence R
description BINDING SITE FOR RESIDUE 3BV Y 301
source : BC7

9) chain Y
residue 20
type
sequence A
description BINDING SITE FOR RESIDUE 3BV Y 301
source : BC7

10) chain Y
residue 21
type
sequence T
description BINDING SITE FOR RESIDUE 3BV Y 301
source : BC7

11) chain Y
residue 33
type
sequence K
description BINDING SITE FOR RESIDUE 3BV Y 301
source : BC7

12) chain Y
residue 47
type
sequence G
description BINDING SITE FOR RESIDUE 3BV Y 301
source : BC7

13) chain Y
residue 49
type
sequence A
description BINDING SITE FOR RESIDUE 3BV Y 301
source : BC7

14) chain Y
residue 170
type
sequence Y
description BINDING SITE FOR RESIDUE 3BV Y 301
source : BC7

15) chain Y
residue 165
type
sequence A
description BINDING SITE FOR RESIDUE MG Y 302
source : BC8

16) chain Y
residue 168
type
sequence D
description BINDING SITE FOR RESIDUE MG Y 302
source : BC8

17) chain Y
residue 169
type
sequence A
description BINDING SITE FOR RESIDUE MG Y 302
source : BC8

18) chain Y
residue 171
type
sequence S
description BINDING SITE FOR RESIDUE MG Y 302
source : BC8

19) chain Y
residue 49
type BINDING
sequence A
description
source Swiss-Prot : SWS_FT_FI2


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